Arylalkyl indoles having serotonin receptor affinity useful...

Drug – bio-affecting and body treating compositions – Designated organic active ingredient containing – Having -c- – wherein x is chalcogen – bonded directly to...

Reexamination Certificate

Rate now

  [ 0.00 ] – not rated yet Voters 0   Comments 0

Details

C514S254080, C514S323000, C548S420000, C546S200000, C544S372000

Reexamination Certificate

active

10518624

ABSTRACT:
The present invention relates to novel tetracyclic arylalkyl indoles, their derivatives, their analogues, their tautomeric forms, their stereoisomers, their polymorphs, their pharmaceutically acceptable salts, their pharmaceutically acceptable solvates, novel intermediates described herein and pharmaceutically acceptable compositions containing them. This invention particularly relates to novel tetracyclic arylalkyl of the general formula (I), their derivatives, their analogues, their tautomeric forms, their stereoisomers, their polymorphs, their pharmaceutically acceptable salts, their pharmaceutically acceptable solvates, novel intermediates described herein and pharmaceutically acceptable compositions containing them. This invention also relates to process/es for preparing such compound/s of general formula (I), composition/s containing effective amount/s of such a compound and the use of such a compound/composition in therapy.

REFERENCES:
patent: 4839377 (1989-06-01), Bays et al.
patent: 4855314 (1989-08-01), Oxford et al.
patent: 303506 (1989-02-01), None
patent: 313397 (1989-04-01), None
patent: 354777 (1991-02-01), None
patent: 438230 (1991-07-01), None
patent: 457701 (1991-11-01), None
patent: 497512 (1992-08-01), None
patent: 2035310 (1980-06-01), None
patent: 91/18897 (1991-12-01), None
patent: 93/00086 (1993-01-01), None
patent: 93/23396 (1993-11-01), None
patent: 94/06769 (1994-03-01), None
Morissette et al. Advanced Drug Delivery Reviews 2004, 56, 275-300.
Kozikowski et al. Tetrahedron Lett. 1991, 32(28), 3317-20.
Barnes et al. Neuropharmacology 1999, 38, 1083-1152.
Bassiony et al. Psychosomatics 2003, 44(5), 388-401.
Gershon, M. D. Ailment Pharmacol. Ther. 2004, 20(suppl. 7), 3-14.
Fuller, R.W., Drugs Acting on Serotonergic Neuronal Systems, Biology of Serotonergic Transmission, John Wiley & Sons Ltd. (1982), 221-247.
Gershon M.D. et al., The periphal actions of 5-Hydroxytryptamine (1989), 246.
Saxena P.R. et al., Journal of Cardiovascular Pharmacology (1990), supplement 7,15.
Glennon et al., Neuroscience and Behavioral Reviews (1990), 14, 35.
Hoyer D. et al., Pharmacol. Rev. (1994), 46, 157-203.
Ruat M. et al., Biochem. Biophys. Res. Com. (1993), 193, 269-276.
Roth et al., J. Pharm. Exp. Therapeut. (1994), 268, 1403-1410.
Sleight et al., Exp. Opin Ther. Patents (1998), 8, 1217-1224.
Bourson et al, Brit J. Pharmacol. (1998), 125, 1562-1566.
Boess et al, Mol. Pharmacol., 1998, 54, 577-583.
Sleight et al., Brit J. Pharmacol. (1998), 124, 556-562.
Yoshioka et al, Life Sciences (1998), 17/18, 1473-1477.
Schoeffter P. et al. “SDZ216-525, a selective and potent 5-HT1A receptor antagonist” European Journal of Pharmacology, 224, 251-257 (1993).

LandOfFree

Say what you really think

Search LandOfFree.com for the USA inventors and patents. Rate them and share your experience with other people.

Rating

Arylalkyl indoles having serotonin receptor affinity useful... does not yet have a rating. At this time, there are no reviews or comments for this patent.

If you have personal experience with Arylalkyl indoles having serotonin receptor affinity useful..., we encourage you to share that experience with our LandOfFree.com community. Your opinion is very important and Arylalkyl indoles having serotonin receptor affinity useful... will most certainly appreciate the feedback.

Rate now

     

Profile ID: LFUS-PAI-O-3855313

  Search
All data on this website is collected from public sources. Our data reflects the most accurate information available at the time of publication.