Aryl- and heteroaryl piperazinyl carboxamides having central ner

Details Aryl- and heteroaryl piperazinyl carboxamides having central ner Aryl- and heteroaryl piperazinyl carboxamides having central ner

1990-03-14

1991-04-23

Shah, Mukund J.

Drug, bio-affecting and body treating compositions

Designated organic active ingredient containing

Heterocyclic carbon compounds containing a hetero ring...

514247, 514253, 544238, 544294, 544295, 544360, 544373, 544376, 544380, A61K 31505, C07D40304, C07D40314

Patent

active

050100785

ABSTRACT:
There are disclosed compounds of the formula (I) ##STR1## wherein R.sup.1 is 1-adamantyl, 3-methyl-1-adamantyl, 3-noradamantyl, unsubstituted or substituted-2-indolyl, 3-indolyl, 2-benzofuranyl and 3-benzofuranyl wherein the substituents are selected from lower alkyl, lower alkoxy and halo; R.sup.2 is unsubstituted or substituted phenyl, benzyl, pyridinyl, pyrimidinyl or pyrazinyl, wherein the substituents are selected from lower alkyl, lower alkoxy, trifluoromethyl and halo; R.sup.3 is H or lower alkyl of 1 to 3 carbon atoms; n is the integer 0 or 1; m is the integer from 2 to 5; and the pharmaceutically acceptable salts thereof.

REFERENCES:
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patent: 3734915 (1973-05-01), Wright
patent: 4001223 (1975-12-01), Sugimoto
patent: 4202898 (1980-05-01), Depoortere
patent: 4748247 (1988-03-01), Abou-Gharbia
patent: 4797489 (1989-01-01), Abou-Gharbia
patent: 4818756 (1989-04-01), Seidel et al.
patent: 4873331 (1989-10-01), Childers et al.
patent: 4880930 (1989-11-01), New
Chemical Abstracts Index Guide 1982-1986, p. 1189G (1987).
Dompert et al, Chemical Abstracts, vol. 102, No. 220896 (1985).

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