Organic compounds -- part of the class 532-570 series – Organic compounds – Amino nitrogen containing
Patent
1997-07-30
2000-01-11
Dees, Jose' G.
Organic compounds -- part of the class 532-570 series
Organic compounds
Amino nitrogen containing
564123, 564160, C07C23900, C07C23700
Patent
active
060138378
DESCRIPTION:
BRIEF SUMMARY
The present invention relates to new aromatic amides, their preparation process, the compositions containing them and their use as pesticides.
Certain 5-cyclopropyl pentadieneamides are described in the European Patent Applications published under the numbers 0,369,762, 0,524,041 and 0,553,081 as having such properties.
It has now been found that the compounds corresponding to formula (I) as defined hereafter also have useful pesticide properties, which make them capable of being used for the protection of plants, safeguarding hygiene in public or private premises, as well as for the implementation of therapeutic treatment for veterinary use, or even for human use.
The products of formula (I) are moreover photostable and not very toxic for mammals and therefore correspond perfectly to the requirements of the modern agrochemical industry.
Therefore a subject of the present invention is in all their stereoisomeric forms or in the form of stereoisomer mixtures, the compounds of formula (I): -C(X.sub.2)--N(R.sub.1)(R.sub.2) (I) hydrocarbon containing a benzene ring, which is linked to an adjacent (CH.sub.2).sub.a group by a carbon atom of said benzene ring, Q contains 6 to 12 carbon atoms and can be either non-substituted or substituted, a and b are identical or different and independently of each other are equal to 0 or to 1, non-substituted or substituted, bicyclic hydrocarbon containing a benzene ring, which is linked to the adjacent Q.sub.1 and C(X.sub.2) groups by two carbon atoms of said benzene ring, Q.sub.2 contains 6 to 12 carbon atoms and can independently of Q, be either non-substituted or substituted, hydrogen atom, aromatic or non-aromatic, cyclic or acyclic hydrocarbon, and containing 1 to 12 carbon atoms, itself being able to be either non-substituted or substituted, or a radical derived from a linear or branched structure containing 1 to 20 carbon atoms and 1 to 6 heteroatoms chosen from oxygen, nitrogen or sulphur atoms, itself being able to be either non-substituted or substituted, or a radical derived from an aromatic or non-aromatic heterocycle containing 5 to 9 carbon atoms and 1 to 4 heteroatoms chosen from oxygen, nitrogen or sulphur atoms, this radical being able to be non-substituted or substituted, or a group (A): ##STR1## in which X.sub.3 represents an oxygen atom or a sulphur atom, and R.sub.3 represents a hydrogen atom or an R.sub.4 -(T.sub.1).sub.i group in which i is equal to 0 or to 1, T.sub.1 represents a bivalent oxy, carbonyl or oxycarbonyl group and R.sub.4 represents a hydrogen atom or a radical derived from a saturated or unsaturated, linear or branched, aromatic or non-aromatic, cyclic or acyclic hydrocarbon, and containing 1 to 20 carbon atoms, itself being able to be either non-substituted or substituted, or a group (B): ##STR2## in which R.sub.3 and X.sub.3 are as defined above, or a group (C): sulphonyloxy radical and R.sub.5 represents an hydrogen atom or a radical derived from a saturated or unsaturated, linear or branched, aromatic or non-aromatic, cyclic or acyclic hydrocarbon, and containing 1 to 8 carbon atoms, itself being able to be either non-substituted or substituted, or a group (D): a hydrogen atom or a radical derived from a saturated or unsaturated, linear or branched, aromatic or non-aromatic, cyclic or acyclic hydrocarbon, and containing 1 to 8 carbon atoms, itself being able to be either non-substituted or substituted, and R.sub.7 represents a carboxy, fluorocarbonyl, alkoxycarbonyl group containing 2 to 5 carbon atoms, or an acyl radical containing 1 to 5 carbon atoms, or an alkyl radical containing 1 to 4 carbon atoms substituted by a cyano group or by an alkoxycarbonyl radical containing 2 to 5 carbon atoms, or an acyl radical containing 1 to 5 carbon atoms, or by an aryl radical containing 6 to 10 carbon atoms, non-substituted or substituted by one or more groups chosen from halo, cyano, nitro, trifluoromethyl, trifluoro-methoxy, trifluoromethylthio groups or alkyl radicals containing 1 to 4 carbon atoms or alkoxy radicals containing 1 to 4 carbon
REFERENCES:
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Demassey Jacques
Gohar Michel
Wehrey Christian
Dees Jos,e G.
Hoechst Marion Roussel
Qazi Sabiha N.
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