Drug – bio-affecting and body treating compositions – Designated organic active ingredient containing – Having -c- – wherein x is chalcogen – bonded directly to...
Patent
1987-10-02
1990-02-06
Schwartz, Richard A.
Drug, bio-affecting and body treating compositions
Designated organic active ingredient containing
Having -c-, wherein x is chalcogen, bonded directly to...
514397, 514398, 548101, 548103, 548110, 548112, 548119, 548301, 548336, 548337, A61K 31415
Patent
active
048988782
ABSTRACT:
Therapeutic antioxidant compounds, useful for relieving the pathogenesis of oxidative stress, of formula ##STR1## wherein substituents R.sub.1, R.sub.2, R.sub.3, and R.sub.4 are individually selected from among hydrogen, methyl, or other atoms and groups that do not adversely affect the overall spectrum of redox activity of the 4-thiohistidine. N-3 is unsubstituted or is substituted as described for R.sub.1 to R.sub.4. R.sub.6 is preferably hydrogen or --SR.
REFERENCES:
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Holler Tod P.
Hopkins Paul B.
Klevit Rachel E.
Shapiro Bennett M.
Spaltenstein Andreas
Schwartz Richard A.
The Board of Regents of the University of Washington
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