Antibody-drug conjugates

Details Antibody-drug conjugates Antibody-drug conjugates

1991-01-22

1996-05-07

Shah, Mukund J.

Organic compounds -- part of the class 532-570 series

Organic compounds

Chalcogen in the nitrogen containing substituent

560 41, 560 49, 560 17, 560 61, 560139, 560153, 560154, 560171, 546 51, 562400, C07D26530

Patent

active

055147941

ABSTRACT:
Derivatized drugs are prepared with a linker consisting of a malonate, wherein the drug is linked through a methylene to the 2-position carbon of the malonate.

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