Antibacterial and/or antiprotozoal nitromidazole derivative...

Details Antibacterial and/or antiprotozoal nitromidazole derivative... Antibacterial and/or antiprotozoal nitromidazole derivative...

2004-10-27

2009-10-27

Anderson, Rebecca L (Department: 1626)

Organic compounds -- part of the class 532-570 series

Organic compounds

Heterocyclic carbon compounds containing a hetero ring...

C514S392000

Reexamination Certificate

active

07608724

ABSTRACT:
The present application describes nitroimidazolic derivative compounds with antibacterial and/or antiprotozoal activity, which are potent urease inhibitors. It also describes the process for preparing those compounds and their use in pharmaceutical compositions and medicines.

REFERENCES:
patent: 4160827 (1979-07-01), Cho et al.
patent: 4456610 (1984-06-01), Hofheinz et al.
patent: 4482722 (1984-11-01), Thorbek et al.
patent: 6271250 (2001-08-01), Yu
patent: 6423707 (2002-07-01), Yang et al.
patent: 1390836 (2003-01-01), None
patent: 1400312 (2003-03-01), None
patent: 330 201 (1989-08-01), None
patent: 1 355 529 (1974-06-01), None
patent: 1453417 (1976-10-01), None
Permentier et al. (CAPLUS abstract, Accession # 1993:81376, Bulletin des Societes Chimiques Belges (1992), 101(8), 701-7).
Vermeersch et al. (CAPLUS Abstract, accession # 1990:526092, International Journal of Pharmaceutics (1990), 60(3), 253-60).
Bundgaard (Design of Prodrugs, (1985), Elsevier, pages included 1-28).
Krogsgaard-Larsen et al. (Textbook of Drug Design and Discovery, (2002), pages included: 428, 456, 457).
Amtul et al. (Current Medicinal Chemistry, 2002, vol. 9, No. 14, p. 1323-48).
Beaman et al., Antimicrobial Agents and Chemotherapy, Vol Date 1967, 1968, pp. 520-530.
Skupin et al., Tetrahedron: Asymmetry, vol. 8, No. 14, 1997, pp. 2453-2464.
Borlinghaus et al., Cancer Research, vol. 47, No. 15, 1987, pp. 4071-4075.
Tian et al., Chinese Journal of Chemistry, vol. 21, No. 7, 2003, pp. 853-857.
Webb et al., Journal of Laelled Compounds and Radiopharmaceuticals, vol. 28, No. 3, 1990, pp. 265-271.
Pfoertner et al., Journal Helvetical Chimica Acta, vol. 70, No. 1, 1987, pp. 171-174.
Woo et al., Arch Pharm Res., vol. 21., No. 1, pp. 6-11, (Feb. 1998). (abstract).
Ito et al., Eur J Phamacol., vol. 345, No. 2, pp. 193-198, (Mar. 19, 1998). (abstract).
Menendez et al., Mutat Res., vol. 478, No. 1-2, pp. 153-158, (Jul. 1, 2001). (abstract).
Cho et al., J Pharm Sci., vol. 8, No. 8, pp. 883-885, (Aug. 1985). (abstract).
Mahfouz et al., J Pharm Pharmacol., vol. 53, No. 6, pp. 841-848, (Jun. 2001). (abstract).
Park et al., Biol Pharm Bull, vol. 19, No. 2, pp. 182-187, (Feb. 1996). (abstract).
Ohta et al., Biochem Biophys Res Commun., vol. 285, No. 3, pp. 728-733, (Jul. 20, 2001). (abstract).
Odake et al., Biol Pharm Bull. vol. 17, No. 10, pp. 1329-1332, (Oct. 1994). (abstract).
Kuhler et al., J Med Chem., vol. 38, No. 25, pp. 4906-4916, (Dec. 8, 1995). (abstract).
Nagata et al., Antimicrobial Agents and Chemotherapy, vol. 39, No. 10, pp. 2187-2192, (Oct. 1995).
Houimel et al., Eur. J. Biochem., vol. 262, pp. 774-780, (1999).
Chung et al., Brazilian Journal of Pharmaceutical Sciences, vol. 41, No. 2, pp. 155-178, (Jun. 2005). Abstract (see p. 174).

Affiliated with

Also associated with

Rating

Antibacterial and/or antiprotozoal nitromidazole derivative... does not yet have a rating. At this time, there are no reviews or comments for this patent.

If you have personal experience with Antibacterial and/or antiprotozoal nitromidazole derivative..., we encourage you to share that experience with our LandOfFree.com community. Your opinion is very important and Antibacterial and/or antiprotozoal nitromidazole derivative... will most certainly appreciate the feedback.

Rate now

Comments { 0 }

Profile ID: LFUS-PAI-O-4143709