Antibacterial agents

Drug – bio-affecting and body treating compositions – Designated organic active ingredient containing – Peptide containing doai

Reexamination Certificate

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C562S621000, C562S623000

Reexamination Certificate

active

07323448

ABSTRACT:
Compounds of formula (I) or a pharmaceutically or veterinarily acceptable salts thereofwherein R1represents hydrogen, C1-C6alkyl or C1-C6alkyl substituted by one or more halogen atoms; R2represents a group R10-(ALK)m-, and A represents (i) a group of formula (IA):wherein the compounds inhibit the activity of bacterial PDF enzyme.

REFERENCES:
patent: 3166587 (1965-01-01), Bernstein et al.
patent: 3692787 (1972-09-01), Roth et al.
patent: 4996358 (1991-02-01), Handa et al.
patent: 5962666 (1999-10-01), Lonetto
patent: 6045795 (2000-04-01), Ulevitch et al.
patent: 6423690 (2002-07-01), Hunter et al.
patent: 6441042 (2002-08-01), Hunter et al.
patent: 6787522 (2004-09-01), Hunter et al.
patent: 6908911 (2005-06-01), Hunter et al.
patent: 33 20 175 (1984-12-01), None
patent: 082088 (1983-06-01), None
patent: 236872 (1987-09-01), None
patent: 863152 (1998-09-01), None
patent: 879879 (1998-11-01), None
patent: WO 94/07527 (1994-04-01), None
patent: WO 94/10990 (1994-05-01), None
patent: WO 95/32944 (1995-12-01), None
patent: WO 96/16027 (1996-05-01), None
patent: WO 97/38705 (1997-10-01), None
patent: WO 98/38179 (1998-09-01), None
Y Jin et al.: “Inhibition stereochemistry of hydroxamate inhibitors for thermolysin”, Bioorganic & Medicinal Chemistry Letters, vol. 8, No. 24, 1998, pp. 3515-3518, XP002106374.
M-C Fournie-Zaluski et al.: “New bidentates as full inhibitors of enkephalin-degrading enzymes: synthesis and analgesic properties” Journal of Medicinal Chemistry, vol. 28, No. 9, 1985, pp. 1158-1169, XP002019770.
H.N. Weller, et al.: “Design of conformality Constrained Angiotensin-Converting Enzyme Inhibitors” Biochemical and Biophysical Research Communications, vol. 125, No. 1, 1984, pp. 82-89, XP002106375.
D. Mazel et al.: “Genetic Characteristics of Polypeptide Deformylase, A Distinctive Enzyme of Eubacterial Translation” EMBO, vol. 13, No. 4, pp. 914-923, XP002043973, (1994).
P.T. Ravi Rajagopalan et al.: “Peptide Deformylas: A New Type of Mononuclear Iron Protein”, JAm.Chem.Soc., vol. 119, 1997, pp. 12418-21419, XP002106376.

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