Drug – bio-affecting and body treating compositions – Designated organic active ingredient containing – Heterocyclic carbon compounds containing a hetero ring...
Reexamination Certificate
2007-05-29
2007-05-29
Owens, Amelia A. (Department: 1625)
Drug, bio-affecting and body treating compositions
Designated organic active ingredient containing
Heterocyclic carbon compounds containing a hetero ring...
C514S313000, C514S314000, C514S315000, C514S316000, C514S318000, C514S248000, C514S256000, C546S184000, C546S187000, C546S159000, C546S152000, C546S170000, C546S192000, C544S182000, C544S194000, C544S198000, C544S238000, C544S242000, C544S256000, C544S297000, C544S322000
Reexamination Certificate
active
10940615
ABSTRACT:
The invention relates to antibacterial 3,5-diaminopiperidine-substituted aromatic and heteroaromatic compounds and pharmaceutical compositions thereof. This invention also relates to a method of using such compounds in the treatment of bacterial infections in mammals, especially humans.
REFERENCES:
patent: 3879790 (1975-04-01), Girard
patent: 4522643 (1985-06-01), Quinlan
patent: 5238936 (1993-08-01), Regnier et al.
patent: 5300643 (1994-04-01), Grohe et al.
patent: 5574055 (1996-11-01), Borgulya et al.
patent: 5852019 (1998-12-01), Ejima et al.
patent: 6248306 (2001-06-01), Schmitt-Willich et al.
patent: 6514977 (2003-02-01), Anantanarayan et al.
patent: 2003/0106169 (2003-06-01), Vidal et al.
patent: 2002338537 (2002-11-01), None
patent: WO-96/04914 (1996-02-01), None
patent: WO-96/28164 (1996-09-01), None
patent: WO-96/32945 (1996-10-01), None
patent: WO-97/18220 (1997-05-01), None
patent: WO-00/056729 (2000-09-01), None
patent: WO-01/10834 (2001-02-01), None
patent: WO-01/023386 (2001-04-01), None
patent: WO-01/023390 (2001-04-01), None
patent: WO-02/056882 (2002-07-01), None
patent: WO-02/060877 (2002-08-01), None
patent: WO-02/078659 (2002-10-01), None
patent: WO-03/059894 (2003-07-01), None
patent: WO-03/101980 (2003-12-01), None
patent: WO-04/002948 (2004-01-01), None
Ames and Ward, “[1,4] Benzodioxinopyridazines,”J. Chem. Soc., 6, 534-538 (1975).
Breshears et al., “The Aminolysis of Certain Chlorosubstituted Purines,”J. Am. Chem. Soc., 81, 3789-3792 (1959).
Elsager et al., “Folate Antagonists, 3. 2,4-Diamino-6-(heterocyclic)quinazolines, a Novel Class of Antimetabolites with Potent Antimalarial and Antibacterial Activity,”J. Med. Chem., 15(8), 827-836 (1972).
Grasa and Nolan, “Palladium/Imidazolium Salt Catalyzed Coupling of Aryl Halides with Hypervalent Organostannates,”Org. Lett., 3(1), 119-122 (2001).
Gujadhur et al., “Formation of Aryl—Nitrogen Bonds Using a Soluble Copper(I) Catalyst,”Tet. Lett., 42, 4791-4793 (2001).
Ji et al., “Selective Amination of Polyhalopyridines Catalyzed by a Palladium-Xantphos Comples,”Organic Letters, 5(24), 4611-4614 (2003).
La Brecque et al., “Substituted Melamines as Chemosterilants of House Flies,”J. Economic Entomology, 61(6), 1621-1632 (1968).
Lebreton et al., “Antibacterial single-bead screening,”Tetrahedron, 59, 10213-10222 (2003).
Littke and Fu, “Palladium-Catalyzed Coupling Reactions of Aryl Chlorides,”Angew. Chem. Int. Ed., 41, 4176-4211 (2000).
Menicagli et al., “in VitroCytotoxic Activities of 2-Alkyl-4,6-diheteroalkyl-1,3,5-triazines: New Molecules in Anticancer Research,”J. Med. Chem., 47, 4649-4652 (2004).
Menichincheri et al., “Parallel Synthesis of 4-Amino-2,6-Dialkylamino-Pyridines,”Tet. Lett., 44, 519-522 (2003).
Ayida Benjamin
Gregor Vlad E.
Hermann Thomas
Murphy Douglas
Simonsen Klaus B.
Anadys Pharmaceuticals, Inc.
Connolly Bove & Lodge & Hutz LLP
Owens Amelia A.
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