Anti-neoplastic, anti-viral or anti-retroviral spermine derivati

Drug – bio-affecting and body treating compositions – Designated organic active ingredient containing – Having -c- – wherein x is chalcogen – bonded directly to...

Patent

Rate now

  [ 0.00 ] – not rated yet Voters 0   Comments 0

Details

514654, 514674, A61K 31505, A61K 31135, A61K 3113

Patent

active

056818378

ABSTRACT:
A mosquito insecticidal composition for controlling the growth of mosquitos wherein the active agent is a polyamine having one of the formulae: ##STR1## wherein: R.sub.1 and R.sub.6 may be the same or different and are alkyl having from 1 to 12 carbon atoms or hydrocarbyl aralkyl having up to 12 carbon atoms;
R.sub.2 -R.sub.5 may be the same or different and are H, R.sub.1 or R.sub.6 ;
R.sub.7 is H, alkyl having from 1 to 12 carbon atoms, hydrocarbyl aryl or hydrocarbyl aralkyl, each having up to 12 carbon atoms;
m is an integer from 3 to 6, inclusive;
n is an integer from 3 to 6, inclusive; or
(IV) a salt thereof with an acid and a carrier therefor.

REFERENCES:
patent: 2267204 (1941-12-01), Kyrides
patent: 2279294 (1942-04-01), Hardman
patent: 2951092 (1960-08-01), Sowinski et al.
patent: 3369905 (1968-02-01), Jones et al.
patent: 3697659 (1972-10-01), Marco
patent: 4010200 (1977-03-01), Kalopissis et al.
patent: 4172094 (1979-10-01), Dybas et al.
patent: 4279621 (1981-07-01), Reusser
patent: 4321190 (1982-03-01), Costanzi et al.
patent: 4505861 (1985-03-01), Bergeron Jr.
patent: 4507321 (1985-03-01), Raisfeld
patent: 4559362 (1985-12-01), Umezawa et al.
patent: 4591605 (1986-05-01), Ray
patent: 5091576 (1992-02-01), Bergeron
patent: 5109024 (1992-04-01), Prakash et al.
patent: 5217964 (1993-06-01), Edwards et al.
patent: 5342945 (1994-08-01), Bergeron
patent: 5393757 (1995-02-01), Bergeron, Jr. et al.
patent: 5434145 (1995-07-01), Edwards et al.
patent: 5455277 (1995-10-01), Bergeron
Niutsu et al, "Synthesis of a Series of Linear Pentamines with Three and Four Methylene Chain Intervals", ChemPharm. Bull, vol. 34(3) 1032-1038, 1986.
Bergeron, "Methods for the Selective Modification of Spermidine and its Homologues", Acc. Chem. Res. 1986, 19, 105-113.
Israel et al, "Synthesis of amino ethyl derivatives of .alpha., .omega.-alkylenediamines and Structure Activity Relationships for the Polyamine-Bovine Plasma Amine Oxadase System", Journal of Medicinal Chemistry, 1971, vol. 14, No. 11, pp. 1042-1047.
Brown et al, "Fungicidal Activity and Chemical Constitution XXI. The Fungitoxity of Alphatic Amines", Pestic. Sci, 1973, 4, 485-490.
Weinstock et al, "Synthesis of Now Polyamine Derivatives for Cancer Chemotherapeutic Studies", Journal of Pharmaceutical Sciences, vol. 70, No Aug. 198.

LandOfFree

Say what you really think

Search LandOfFree.com for the USA inventors and patents. Rate them and share your experience with other people.

Rating

Anti-neoplastic, anti-viral or anti-retroviral spermine derivati does not yet have a rating. At this time, there are no reviews or comments for this patent.

If you have personal experience with Anti-neoplastic, anti-viral or anti-retroviral spermine derivati, we encourage you to share that experience with our LandOfFree.com community. Your opinion is very important and Anti-neoplastic, anti-viral or anti-retroviral spermine derivati will most certainly appreciate the feedback.

Rate now

     

Profile ID: LFUS-PAI-O-1026244

  Search
All data on this website is collected from public sources. Our data reflects the most accurate information available at the time of publication.