Anti-inflammatory glucocorticoid compounds for topical ophthalmi

Drug – bio-affecting and body treating compositions – Designated organic active ingredient containing – Cyclopentanohydrophenanthrene ring system doai

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514174, 514175, 514176, 540 2, 540 67, 540108, 540111, 540115, 540116, 540118, 540120, A61K 3158, C07J 3100, C07J 4300, C07J 3300

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active

054201209

ABSTRACT:
Topically administrable C-21 thioether glucocorticoid steroid derivatives are disclosed as effective anti-inflammatory agents for the treatment of ophthalmic inflammatory disorders. These C-21 thioether derivatives do not cause a significant increase in intraocular pressure as a side effect.

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