Drug – bio-affecting and body treating compositions – Designated organic active ingredient containing – Heterocyclic carbon compounds containing a hetero ring...
Patent
1991-08-12
1993-05-04
Robinson, Allen J.
Drug, bio-affecting and body treating compositions
Designated organic active ingredient containing
Heterocyclic carbon compounds containing a hetero ring...
514183, 5142312, 5142388, A61K 3133, A61K 31535
Patent
active
052082334
ABSTRACT:
There are disclosed anti-hypertensive compositions and a method of lowering blood pressure in mammals. The active component in the anti-hypertensive compositions is a compound of the formula ##STR1## wherein R.sub.1 and R.sub.2 are independently selected from straight chain and branched chain C.sub.1 -C.sub.12 alkyl groups and benzyl, with the proviso that no branch occur on the alpha carbon atom of the alkyl group; or R.sub.1 and R.sub.2 together with the nitrogen atom they are bonded to form a heterocyclic ring; M.sup.+X is a pharmaceutically acceptable cation, wherein x is the valence of the cation.
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Dunams Tambra M.
Hrabie Joseph A.
Keefer Larry K.
Wink David A.
Robinson Allen J.
The United States of America as represented by the Department of
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