Drug – bio-affecting and body treating compositions – Designated organic active ingredient containing – Having -c- – wherein x is chalcogen – bonded directly to...
Patent
1990-11-28
1992-09-29
Shah, Mukund J.
Drug, bio-affecting and body treating compositions
Designated organic active ingredient containing
Having -c-, wherein x is chalcogen, bonded directly to...
514241, 514242, 514243, 514248, 514249, 514252, 514259, 544182, 544183, 544219, 544238, 544284, 544296, 544295, 544319, A61K 31505, C07D239545
Patent
active
051514273
ABSTRACT:
Novel anthelmintics are described which, as active ingredient, contain a compound of the formula I ##STR1## or in its hydrogenated form the formula (Ia) ##STR2## in which R.sub.1 and R.sub.2 independently of one another are C.sub.1 -C.sub.6 alkyl, allyl, C.sub.3 -C.sub.6 cycloalkyl, benzyl or phenyl; R.sub.3 is an unsubstituted or substituted heteroaromatic 6-membered ring which contains 1, 2 or 3 nitrogen atoms or a benzo-fused, unsubstituted or substituted heteroaromatic 6-membered ring which contains 1 to 3 nitrogen atoms, and R.sub.4 and R.sub.5 independently of one another are hydrogen, C.sub.1 -C.sub.4 alkyl, C.sub.1 -C.sub.4 alkoxy or halogeno-C.sub.1 -C.sub.3 alkyl, including their tautomeric forms and physiologically tolerable salts. The preparation, formulation and use of these active ingredients are also described.
REFERENCES:
patent: 4602912 (1986-07-01), deSousa et al.
patent: 4636508 (1987-01-01), Brewer et al.
patent: 4670441 (1987-06-01), Kuhne et al.
patent: 4748178 (1988-05-01), Burkhardt et al.
patent: 4753940 (1988-06-01), Sturm et al.
patent: 4879276 (1989-11-01), Brewer et al.
Chem. Abstr. 103: 215, 248, Mikhavela et al., from Khimgs., (1985), 378-85.
Chem. Abstr: 113:6366, Brewer et al., Abstr. from South African Patent 88 03, 119 (Sep. 1989).
Chem Abstr. 112:139,048, Brewer et al., From BE 1,001,262 (Sep. 1989).
Chem Abstr. 112:198,414, Brewer et al., from FR 2,628,869 (Sep. 1989).
Chem Abstr. 112:118,846, Brewer et al., from BE 1,001,263 (Sep. 1989).
Chem Abstr. 111:225,323, Warrell et al., from WO 8810,114 (Jun. 1987).
G. W. Benz et al., Amer. J. Vet Res., 38, pp. 1425-1426 (1976).
V. J. Theodorides et al., Amer. J. Vet. Res., 37, 1515-1516 (1976).
R. A. Knight et al., Amer. J. Vet. Res., 38, 807-808 (1976).
H. Herlick, Amer. J. Vet. Res., 38 pp. 1247-1248 (1977).
Ciba-Geigy Corporation
Grumbling Matthew V.
Mathias Marla J.
Roberts McC. Edward
Shah Mukund J.
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