Chemistry of carbon compounds – Miscellaneous organic carbon compounds – C-metal
Patent
1975-08-19
1977-05-17
Daus, Donald G.
Chemistry of carbon compounds
Miscellaneous organic carbon compounds
C-metal
260DIG8, 260285, 424250, C07D47108
Patent
active
040240827
ABSTRACT:
dl-N-Cyclopropylmethyl-3-hydroxy-9-azamorphinan is a compound known to possess analgesic activity that is about twice as potent as pentazocine. Resolution of the compound into its levorotatory and dextrorotatory isomers and subsequent animal testing revealed that l-N-cyclopropylmethyl-3-hydroxy-9-azamorphinan was much more potent than the dl-mixture.
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Gordon Maxwell
Kametani Tetsuji
Kigasawa Kazuo
Partyka Richard Anthony
Berch Mark L.
Bristol-Myers Company
Daus Donald G.
Lloyd Richard R.
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