Aminopropylphosphinic acids

Details Aminopropylphosphinic acids Aminopropylphosphinic acids

2005-01-11

2005-01-11

Richter, Johann (Department: 1621)

Organic compounds -- part of the class 532-570 series

Organic compounds

Phosphorus acids or salts thereof

C562S008000, C514S075000, C514S114000

Reexamination Certificate

active

06841698

ABSTRACT:
Novel compounds of formula I, with the exception ofi) the racemate of (3-amino-2-hydroxypropyl)phosphinic acid; andii) (2R/S,3R)-(3-amino-2-hydroxybutyl)phosphinic acid,having affinity to one or more GABABreceptors, their pharmaceutically acceptable salts, solvates and stereoisomers, as well as processes for their preparation, pharmaceutical compositions containing said therapeutically active compounds and the use of said active compounds in therapy.

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