Aminoalkylbenzofurans as serotonin (5-HT(2c)) agonists

Drug – bio-affecting and body treating compositions – Designated organic active ingredient containing – Having -c- – wherein x is chalcogen – bonded directly to...

Reexamination Certificate

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Details

C514S466000, C514S337000, C549S467000, C546S284100

Reexamination Certificate

active

07045545

ABSTRACT:
The present invention provides serotonergic aminoalkylbenzofurans of Formula (I): where R, R1, R2, R3, R4, R4′, R5, R5′, and R12are as described in the specification.

REFERENCES:
patent: WO 94 29290 (1994-12-01), None
patent: WO 97 08167 (1997-03-01), None
patent: WO 97 43272 (1997-11-01), None
Schulze-Alexandru, M. et al ‘Quasi-atomistic receptor surrogates for the 5-HT2A receptor: a 3D-QSAR study on hallucinogenic substances’ CA 132:202636 (2000).
Ellis, F. et al ‘Benzofurans and benzopyrans as chronobiological agents’ CA 128:22811 (1997).
Royer, R. et al ‘Benzofurans. L. Access to furoisoquinolines’ CA 78:71948 (1973).
Wolff, M C et al The discriminative stimulus properties of LY233708, a selective seratonin reuptake inhibitor, in the pigeon, Psychopharmacology, (1999) 146:275-279.
H. Ishii, et al. “Total Synthesis of Lemaireocereine” Chem. Pharm. vol. 40, No. 8, 1992, pgs 1993-1996, XP00887200 p. 1994.
R. Royer, et al. “Recherches Sur le benzofuranne. L.—Étude de voies d'accés aux furoisoquinoléines” Bull. Soc. Chim. Fr., No. 11, 1972,m pp. 4201-4208, XP000088692 table VI.
Schulze-Alexandru, M., et al., n “Quasi-atomistic receptor surrogates for the 5-HT2A receptor: a 3D-QSAR study on hallucinogenic substances” CA 132:202636 (2000).
Ellis, F., et al. “Benzofurans and benzopyrans as chronobiological agents” CA 128:22811 (1997).
Royer, R., et al. “Benzofurans, L. Access to furoisoquinolines” CA 78:71948 (1973).

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