Organic compounds -- part of the class 532-570 series – Organic compounds – Heterocyclic carbon compounds containing a hetero ring...
Reexamination Certificate
2008-07-15
2008-07-15
Seaman, D. Margaret (Department: 1625)
Organic compounds -- part of the class 532-570 series
Organic compounds
Heterocyclic carbon compounds containing a hetero ring...
C564S306000
Reexamination Certificate
active
07399863
ABSTRACT:
The invention provides novel β2adrenergic receptor agonist compounds. The invention also provides pharmaceutical compositions comprising such compounds, methods of using such compounds to treat diseases associated with β2adrenergic receptor activity, and processes and intermediates useful for preparing such compounds.
REFERENCES:
patent: 3875233 (1975-04-01), Bastian et al.
patent: 4021485 (1977-05-01), Schromm et al.
patent: 4894219 (1990-01-01), Baker et al.
patent: 4992474 (1991-02-01), Skidmore et al.
patent: 5223614 (1993-06-01), Schromm et al.
patent: 5434304 (1995-07-01), Trofast et al.
patent: 5750701 (1998-05-01), Beeley et al.
patent: 6268533 (2001-07-01), Gao et al.
patent: 6541669 (2003-04-01), Moran et al.
patent: 6576793 (2003-06-01), Moran et al.
patent: 6653323 (2003-11-01), Moran et al.
patent: 6670376 (2003-12-01), Moran et al.
patent: 6747043 (2004-06-01), Moran et al.
patent: 6759398 (2004-07-01), Biggadike
patent: 6825220 (2004-11-01), Jesudason et al.
patent: 2002/0019378 (2002-02-01), Angell et al.
patent: 2002/0022625 (2002-02-01), Walland et al.
patent: 2002/0143034 (2002-10-01), Taniguchi et al.
patent: 2003/0229058 (2003-12-01), Moran et al.
patent: 2004/0059116 (2004-03-01), Moran et al.
patent: 2004/0063755 (2004-04-01), Moran et al.
patent: 2004/0157830 (2004-08-01), Biggadike et al.
patent: 2004/0180876 (2004-09-01), Biggadike et al.
patent: 2004/0186080 (2004-09-01), Moran et al.
patent: 2004/0224982 (2004-11-01), Axt et al.
patent: 2004/0242890 (2004-12-01), Coe et al.
patent: 2004/0248985 (2004-12-01), Stergiades et al.
patent: 2005/0272769 (2005-12-01), Linsell
patent: 849 794 (1977-04-01), None
patent: 550 768 (1972-02-01), None
patent: 0 233 686 (1987-08-01), None
patent: 0147 719 (1989-07-01), None
patent: 0 196 849 (1996-10-01), None
patent: 1040724 (1966-09-01), None
patent: 52-83379 (1977-07-01), None
patent: 52-83619 (1977-07-01), None
patent: WO 99/64035 (1999-12-01), None
patent: WO 00/75114 (2000-12-01), None
patent: WO 01/42193 (2001-06-01), None
patent: WO 03/024439 (2003-03-01), None
patent: WO 03/042160 (2003-05-01), None
patent: WO 03/042164 (2003-05-01), None
patent: WO 03/072539 (2003-09-01), None
patent: WO 03/091204 (2003-11-01), None
patent: WO 2004/016578 (2004-02-01), None
U.S. Appl. No. 11/033,198, filed Jan. 11, 2005, McKinnell et al.
U.S. Appl. No. 10/627,555, filed May 8, 2003, Linsell et al.
Bompart et al., “Synthesis of new β-blocking analogs of bevantolol”, Annales Pharmaceutiques Francaises, Volume Date 1984, 42(6), pp. 537-545 (1985) (In French with English abstract).
Bompart et al., “Synthesis of new β-blocker analogs of bevantolol or alprenolol”, Annales Pharmaceutiques Francaises, Volume Date 1987, 45(5), pp. 379-387 (1988) (In French with English abstract).
Deyrup et al., “Structure-affinity profile of 8-hydroxycarbostyril-based agonists that dissociate slowly from the Beta2-adrenoceptor”, Naunyn-Schmiedeberg's Arch Pharmacol (1999) 359:168-177.
Isogaya et al., “Binding Pockets of the β1- and β2-Adrenergic Receptors for Subtype-Selective Agonists”), Molecular Pharmacology, vol. 56, pp. 875-885 (1999).
Milecki et al., “Carbostyril Derivatives Having Potent β-Adrenergic Agonist Properties”, J. Med. Chem, (1987), 30, 1563-1566.
Yokoi et al., “The Development of a Radioimmunoassay for Formoterol”, Life Sciences, (1983) vol. 33, No. 17, pp. 1665-1672.
Yoshizaki et al., “Sympathomimetic Amines Having a Carbostyril Nucleus”, J. Med. Chem., (1976), vol. 19, No. 9, pp. 1138-1142.
Office Action in U.S. Appl. No. 10/431,762, dated Apr. 17, 2006.
Office Action in U.S. Appl. No. 10/431,762, dated Sep. 26, 2006.
Office Action in U.S. Appl. No. 10/431,762, dated Mar. 14, 2007.
Jacobsen John R.
Linsell Martin S.
Saito Daisuke Roland
Hagenah Jeffrey A.
Saxon Roberta P.
Seaman D. Margaret
Theravance Inc.
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