Amino-protected dopa derivative and production thereof

Details Amino-protected dopa derivative and production thereof Amino-protected dopa derivative and production thereof

1990-08-17

1992-03-24

Dees, Jose G.

Organic compounds -- part of the class 532-570 series

Organic compounds

Carboxylic acid esters

560 27, 560134, 560163, 560170, 544 1, C07C26900, C07C27100, C07D25300

Patent

active

050989995

ABSTRACT:
3,4-Dihydroxyphenylalanine wherein the amino group is protected with a 9-fluorenylmethyloxycarbonyl group, or a derivative thereof can be produced by reacting 3,4-dihydroxyphenylalanine with a boron compound or phosphorus compound to stabilize the hydroxyl groups, followed by introduction of a 9-fluorenylmethyloxycarbonyl group thereinto.

REFERENCES:
patent: 3846476 (1974-11-01), Kaiser et al.
patent: 3852338 (1974-12-01), Kaiser et al.
patent: 3859331 (1975-01-01), Kaiser et al.
patent: 4311706 (1982-01-01), Bodor et al.
Carpino et al., J. Org. Chem., vol. 37, No. 22, pp. 3404-3409 (1972).
Meienhofer et al., Int. J. Peptide Protein Res., vol. 13, pp. 35-42, (1979).
R. C. de L. Milton et al., Int. J. Peptide Protein Res., vol. 30, pp. 431-432 (1987).
Schon et al., Synthesis, vol. 4, pp. 303-305 (1986).
Chang et al., Int. J. Peptide Protein Res., vol. 15, pp. 59-66 (1980).

Affiliated with

Also associated with

Rating

Amino-protected dopa derivative and production thereof does not yet have a rating. At this time, there are no reviews or comments for this patent.

If you have personal experience with Amino-protected dopa derivative and production thereof, we encourage you to share that experience with our LandOfFree.com community. Your opinion is very important and Amino-protected dopa derivative and production thereof will most certainly appreciate the feedback.

Rate now

Comments { 0 }

Profile ID: LFUS-PAI-O-2011384