Drug – bio-affecting and body treating compositions – Designated organic active ingredient containing – Having -c- – wherein x is chalcogen – bonded directly to...
Patent
1995-06-07
1998-05-26
Richter, Johann
Drug, bio-affecting and body treating compositions
Designated organic active ingredient containing
Having -c-, wherein x is chalcogen, bonded directly to...
514322, 514321, 514319, 514323, 514324, 514326, 514331, 5142372, 5142278, 514252, 514367, 514375, 514394, 514428, 546199, 546198, 546197, 546233, 544 586, 544 585, 544130, 544141, 544360, 544372, A61K 3140, C07D20706
Patent
active
057565333
ABSTRACT:
Selected amino acid hydroxyethylamino sulfonamide compounds are effective as retroviral protease inhibitors, and in particular as inhibitors of HIV protease. The present invention relates to such retroviral protease inhibitors and, more particularly, relates to selected novel compounds, composition and method for inhibiting retroviral proteases, such as human immunodeficiency virus (HIV) protease, prophylactically preventing retroviral infection or the spread of a retrovirus, and treatment of a retroviral infection.
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Brown David L.
DeCrescenzo Gary A.
Devadas Balekudru
Freskos John N.
Getman Daniel P.
Cross Lutz Laura
G.D. Searle & Co.
Richter Johann
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