Amine derivatives of oxo- and hydroxy- substituted hydrocarbons

Details Amine derivatives of oxo- and hydroxy- substituted hydrocarbons Amine derivatives of oxo- and hydroxy- substituted hydrocarbons

1997-07-25

1999-08-24

Shah, Mukund J.

Drug, bio-affecting and body treating compositions

Designated organic active ingredient containing

Heterocyclic carbon compounds containing a hetero ring...

514247, 514248, 514252, 514253, 514311, 540553, 544237, 544238, 546169, C07D21548, A61K 3147

Patent

active

059425040

ABSTRACT:
The present invention discloses the compounds of general formula (1) ##STR1## wherein R.sup.1, R.sup.2, R.sup.3 are optionally substituted carbonyl and amide derivatives which are useful as inhibitors of retroviral proteases, and are effective in treating conditions characterized by unwanted activity of these enzymes, such as acquired immune deficiency syndrome.

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