Amidino compounds as cysteine protease inhibitors

Details Amidino compounds as cysteine protease inhibitors Amidino compounds as cysteine protease inhibitors

2004-06-04

2010-02-16

Chang, Celia (Department: 1625)

Drug, bio-affecting and body treating compositions

Designated organic active ingredient containing

Having -c-, wherein x is chalcogen, bonded directly to...

C514S238500, C514S311000, C514S331000, C514S394000, C514S416000, C514S451000, C514S520000, C544S059000, C544S163000, C546S134000, C546S230000, C546S286000, C548S304400, C548S505000, C548S559000, C549S013000, C549S426000, C558S392000

Reexamination Certificate

active

07662849

ABSTRACT:
The present invention is directed to compounds that are inhibitors of cysteine proteases, in particular, cathepsins B, K, L, F, and S and are therefore useful in treating diseases mediated by these proteases. The present invention is directed to pharmaceutical compositions comprising these compounds and processes for preparing them.

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