Amidine and isothiourea derivatives as inhibitors of nitric oxid

Details Amidine and isothiourea derivatives as inhibitors of nitric oxid Amidine and isothiourea derivatives as inhibitors of nitric oxid

1999-01-20

2000-10-31

Shah, Mukund J.

Drug, bio-affecting and body treating compositions

Designated organic active ingredient containing

Heterocyclic carbon compounds containing a hetero ring...

514214, 514215, 514220, 514221, 540558, 540559, 540560, 540561, 540562, 540569, 540570, 540571, 540572, 540573, C07D40912, C07D47104, C07D48904, A61K 31445

Patent

active

061403229

ABSTRACT:
There are provided novel compounds of formula (I) ##STR1## wherein X, R.sup.1, R.sup.2, R.sup.3, R.sup.4 and R.sup.5 are as defined in the specification and optical isomers and racemates thereof and pharmaceutically acceptable salts thereof; together with processes for their preparation, compositions containing them and their use in therapy.

REFERENCES:
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CAS Registry nos. cited against Claim 24:107393-74-8; 102599-10-0; 72299-68-4; 72299-67-3; 72232-26-9; 72232-25-8; 37481-24-6; 14788-34-2; 14097-41-7; 14097-40-6; and 14097-37-1.
CAS Registry nos. cited against Claim 26; 135043-75-3; 135007-64-6; 135007-60-2; 114166-30-2; 114166-29-9; 114166-17-5; 99365-69-2; 69062-43-7; 42923-79-5; 41959-45-9; 14097-36-0; and 14097-35-9.
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