Amides and esters containing bridged piperidines and use as sero

Drug – bio-affecting and body treating compositions – Designated organic active ingredient containing – Having -c- – wherein x is chalcogen – bonded directly to...

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546112, 546183, A61K 31445, C07D40112, C07D40512, C07D22122

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active

047974060

ABSTRACT:
The dicarboxylic, heterocyclic and substituted benzoic acid alkylene bridged piperidyl amides and esters are serotonin M antagonists.

REFERENCES:
patent: 2748134 (1956-05-01), Stoll et al.
patent: 3170927 (1965-02-01), Nador et al.
patent: 3342826 (1967-09-01), Miller et al.
patent: 3405134 (1968-10-01), Judd
patent: 3702324 (1972-11-01), Skinner et al.
patent: 3741973 (1973-06-01), Fonken et al.
patent: 4089960 (1978-05-01), Gosteli et al.
patent: 4093734 (1978-06-01), Kruger et al.
patent: 4213983 (1980-07-01), Hadley et al.
patent: 4273778 (1981-06-01), Hadley et al.
patent: 4459300 (1984-07-01), Watts
patent: 4499099 (1985-02-01), Watts
Chem. Abs. 82:156533e (1975).
Seiler, N., et al., Hoppe-Seyler's Z. Physiol. Chem., vol. 348, 768-774 (1967).
Singh, S., et al., J. Heterocyclic Chem., 16, 625 (1979).
Waters, J., Journal of Med. Chem., vol. 21, No. 7, pp. 628-633 (1978).
Cheng, C., et al., Journal of Med. Chem., vol. 25, No. 2, pp. 145-152 (1982).
Schultz, O., et al., Pharm. Zeit., No. 40, pp. 1455 and 1456.
Derwent Abstract of S. Africa 62/3640 (2/13/63).
Kasztreiner, E., et al., Acta Chim. Acad. Scien. Hung., vol. 51, pp. 327-338 (1967).
Izv. Akad. Nauk. Arm. SSR, Biol. Nauk., vol. 15, No. 12, pp. 3-14 (1962).
Chem. Abs. 59:5665g (1963).
Feher, O., et al., Acta Biologica Szeged., vol. 21, pp. 113-125 (1975).
Chem. Abs. 86:83522w (1977).
Bosse, J., et al., Naunyn-Schmiedebergs Arch. Pharmacol Exp. Path., vol. 259, pp. 34-44 (1967).
House H., et al., J. of Org. Chem., vol. 31, pp. 3482-3489 (1966).
Ohki, E., et al., Chem. Pharm. Bull., vol. 18, No. 10, pp. 2050-2057 (1970).
Mikhlina, E., et al., Khim.-Farm. Zh., vol. 7, No. 8, pp. 492-496 (1973).
Lieberman, H., et al., J. of Pharm. Sciences, vol. 57, pp. 684 and 685 (1968).
Chem. Abs. 54:22632h (1960).
Proceedings of the B.P.S., pp. 499 and 500 (Sep. 7th-9th, 1977), Fozard, J., et al.

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