Drug – bio-affecting and body treating compositions – Designated organic active ingredient containing – Having -c- – wherein x is chalcogen – bonded directly to...
Patent
1995-03-10
1997-04-22
Shah, Mukund J.
Drug, bio-affecting and body treating compositions
Designated organic active ingredient containing
Having -c-, wherein x is chalcogen, bonded directly to...
514422, 514469, 5142335, 514212, 206828, 546196, 544153, 548525, 540596, 549467, A61K 3134, A61K 31445, C07D40510, C07D30780
Patent
active
056229747
ABSTRACT:
This invention relates to the fields of pharmaceutical and organic chemistry and provides novel 3-benzyl-benzofurans which are .alpha.-substituted with ether, thioether amino, cyano or halo that are useful for the treatment of the various medical indications associated with post-menopausal syndrome, as well as estrogen dependent diseases including cancer of the breast, uterus and cervix. The present invention further relates to intermediate compounds and processes useful for preparing the pharmaceutically active compounds of the present invention, and pharmaceutical compositions.
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Durani, et al, Journal of Medical Chemistry, vol. 32, No. 8, Aug. 1989, pp. 1700-1707.
Eli Lilly and Company
Page Kathleen R. S.
Sales James J.
Shah Mukund J.
Strode Janelle D.
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