Alpha-morpholino ribonucleoside derivatives and polymers thereof

Organic compounds -- part of the class 532-570 series – Organic compounds – Four or more ring nitrogens in the bicyclo ring system

Patent

Rate now

  [ 0.00 ] – not rated yet Voters 0   Comments 0

Details

544123, C07D41304, C07D47302, C07D47326

Patent

active

053788419

ABSTRACT:
Alpha-morpholino subunits and polymer compositions composed of alpha-morpholino subunits are disclosed. These subunits can be linked together by uncharged linkages, one to three atoms in length, joining the morpholino nitrogen of one subunit to the 5' exocyclic carbon of an adjacent subunit. Each subunit contains a purine or pyrimidine base-pairing moiety effective to bind by hydrogen bonding to a specific base or base-pair in a target polynucleotide. The polymers of the instant invention can be used in place of standard RNA or DNA oligomers. For example, the target-specific polymers of the invention can be used in a variety of diagnostic assays for detection of RNA or DNA having a given target sequence. Further, the polymers of the invention also have potential use as therapeutic agents.

REFERENCES:
patent: 5034506 (1991-07-01), Summerton et al.
patent: 5142047 (1992-08-01), Summerton et al.
patent: 5185444 (1993-02-01), Summerton et al.
patent: 5217866 (1993-06-01), Summerton et al.
Uchiyama et al., Chemical Abstract 112:139741s (1990), Abstract for JP 01, 172,384 (Jul. 7, 1989).
Stirchak, Nucleic Acids Research, vol. 17, No. 15 (1989), pp. 6129-6141.

LandOfFree

Say what you really think

Search LandOfFree.com for the USA inventors and patents. Rate them and share your experience with other people.

Rating

Alpha-morpholino ribonucleoside derivatives and polymers thereof does not yet have a rating. At this time, there are no reviews or comments for this patent.

If you have personal experience with Alpha-morpholino ribonucleoside derivatives and polymers thereof, we encourage you to share that experience with our LandOfFree.com community. Your opinion is very important and Alpha-morpholino ribonucleoside derivatives and polymers thereof will most certainly appreciate the feedback.

Rate now

     

Profile ID: LFUS-PAI-O-2212578

  Search
All data on this website is collected from public sources. Our data reflects the most accurate information available at the time of publication.