Organic compounds -- part of the class 532-570 series – Organic compounds – Heterocyclic carbon compounds containing a hetero ring...
Patent
1995-03-09
1999-07-06
Davis, Zinna Northington
Organic compounds -- part of the class 532-570 series
Organic compounds
Heterocyclic carbon compounds containing a hetero ring...
C07D20904
Patent
active
059199490
ABSTRACT:
.alpha.-Hydroxy acid esters of formula ##STR1## wherein R2 is lower-alkyl, useful as intermediates in the production of .beta.-aminoalcohols.
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D'Aniello et al., "A Stereoselective Method for the Preparation of HIV-1 Protease Inhibitors Based on the Lewis Acid Mediated Reaction of Allylsilanes and N-Boc-.alpha.-amino", J. Org. Chem. 57:5247-5250 (1992).
Ghosh et al, "3-Tetrahydrofuran and Pyran Urethanes as High-Affinity P.sub.2 -Ligands for HIV-1 Protease Inhibitors", J. Med. Chem. 36:292-294 (1993).
Davis Zinna Northington
Hoffmann-La Roche Inc.
Johnston George W.
Tramaloni Dennis P.
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