Drug – bio-affecting and body treating compositions – Designated organic active ingredient containing – Having -c- – wherein x is chalcogen – bonded directly to...
Reexamination Certificate
2007-09-04
2007-09-04
Shameem, Golam M. M. (Department: 1626)
Drug, bio-affecting and body treating compositions
Designated organic active ingredient containing
Having -c-, wherein x is chalcogen, bonded directly to...
C548S215000, C548S225000, C548S229000, C514S374000
Reexamination Certificate
active
10937187
ABSTRACT:
The present invention relates to acyloxymethylcarbamate oxazolidinones. The compounds of the present invention have potent activity with excellent oral bioavailability against Gram-positive and Gram-negative bacteria.
REFERENCES:
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Mulvihilli, Mark J., et. al., “Synthesis and Application of Novel Glyoxylate-derived Chloroformates,” Synthesis, 2002, pp. 365-370.
Rautio, Jarkko, et. al., “Synthesis and In Vitro Evaluation of Aminoacyloxyalkyl Esters of 2-(6-methoxy-2-naphthyl) propionic Acid as Novel Naproxen Prodrugs for Dermal Drug Delivery,” Pharmaceutical Research, vol. 16, No. 8, 1999, pp. 1172-1178.
Wheeler, W.J., et. al., Journal of Medicinal Chemistry, vol. 22, No. 6, 1979, pp. 657-661.
Boyer Frederick Earl
Choy Allison Laura
Gadwood Robert C.
Josyula Vara Prasad Venkata Nagendra
Kim Ji-Young
Pfizer Inc
Shameem Golam M. M.
Tebbutt Jason G.
Zelson Steve
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