Acylated piperazine derivatives as melanocortin-4 receptor...

Drug – bio-affecting and body treating compositions – Designated organic active ingredient containing – Heterocyclic carbon compounds containing a hetero ring...

Reexamination Certificate

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C514S252110, C514S252130, C514S252140, C514S253050, C514S253060, C514S253090, C514S254010, C514S254020, C514S254030, C514S254050, C514S254100, C514S254100, C544S182000, C544S238000, C544S297000, C544S322000, C544S360000, C544S363000, C544S365000, C544S366000, C544S367000, C544S369000, C544S370000, C544S371000, C544S372000, C544S379000

Reexamination Certificate

active

10788859

ABSTRACT:
Certain novel N-acylated piperazine derivatives are agonists of the human melanocortin receptor(s) and, in particular, are selective agonists of the human melanocortin-4 receptor (MC-4R). They are therefore useful for the treatment, control, or prevention of diseases and disorders responsive to the activation of MC-4R, such as obesity, diabetes, sexual dysfunction, including erectile dysfunction and female sexual dysfunction.

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