Acylated benzylglycosides as inhibitors of smooth muscle cell pr

Details Acylated benzylglycosides as inhibitors of smooth muscle cell pr Acylated benzylglycosides as inhibitors of smooth muscle cell pr

1995-10-20

1998-06-30

Peselev, Elli

Drug, bio-affecting and body treating compositions

Designated organic active ingredient containing

Carbohydrate doai

514 53, 536 172, 536 179, A61K 3170, C07H 1700

Patent

active

057734208

ABSTRACT:
This invention relates to acylated benzylglycosides and a method for their use as smooth muscle cell proliferation inhibitors and as therapeutic compositions for treating diseases and conditions which are characterize by excessive smooth muscle proliferation, such as restenosis. The acylated benzylglycosides of this invention are those of formula I, below: ##STR1## wherein X is ##STR2## R.sup.1 is H, alkyl having 1 to 6 carbon atoms, chloro, bromo, or alkoxy having 1 to 6 carbon atoms;

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