Drug – bio-affecting and body treating compositions – Designated organic active ingredient containing – Having -c- – wherein x is chalcogen – bonded directly to...
Patent
1998-10-27
2000-04-18
Morris, Patricia L.
Drug, bio-affecting and body treating compositions
Designated organic active ingredient containing
Having -c-, wherein x is chalcogen, bonded directly to...
514183, 548101, 5482642, 5482644, A01N 43653, C07D24912
Patent
active
060515929
DESCRIPTION:
BRIEF SUMMARY
The present invention relates to novel acyl-mercapto-triazolyl derivatives, to a process for their preparation and to their use as microbicides.
It is already known that numerous triazolyl derivatives have fungicidal properties (cf. EP-A 0 015 756, EP-A 0 040 345, EP-A 0 052 424, EP-A 0 061 835, EP-A 0 297 345. EP-A 0 094 564, EP-A 0 196 038, EP-A 0 267 778, EP-A 0 378 953Ad, EP-A 0 044 605. EP-A 0 069 442, EP-A 0 055 833, EP-A 0 301 393, DE-A 2 324 010, DE-A 2 737 489, DE-A 2 551 560, EP-A 0 065 485, DE-A 2 735 872, EP-A 0 234 242, DE-A 2 201 063, EP-A 0 145 294 and DE-A 3) 721 786). The activity of these substances is good, but in some cases leaves something to be desired at low application rates.
This invention, accordingly, provides novel acyl-mercapto-triazolyl derivatives of the formula ##STR1## in which R represents alkyl, halogenoalkyl, optionally substituted aryl, optionally, substituted aralkyl, alkoxy, alkylamino or optionally substituted arylamino and ##STR2## R.sup.2 and R.sup.3 are identical or different and each represent optionally substituted alkyl, optionally substituted alkenyl, optionally substituted cycloalkyl, optionally substituted aralkyl, optionally substituted aralkenyl, optionally substituted aroxyalkyl, optionally substituted aryl or optionally substituted heteroaryl, ##STR3## R.sup.4 represents alkyl having 1 to 4 carbon atoms, halogenoalkyl having 1 to 4 carbon atoms and 1 to 5 halogen atoms, optionally halogen-substituted cycloalkyl having 3 to 7 carbon atoms, naphthyl or phenyl which is optionally mono- to trisubstituted bid identical or different substituents selected from the group consisting of halogen, nitro, phenyl, phenoxy alkyl having 1 to 4 carbon atoms, alkoxy having 1 to 4 carbon atoms, halogenoalkyl having 1 to 4 carbon atoms and 1 to 5 halogen atoms, halogenoalkoxy having 1 to 4 carbon atoms and 1 to 5 halogen atoms and halogenoalkylthio having 1 to 4 carbon atoms and 1 to 5 halogen atoms, and identical or different substituents selected from the group consisting of halogen, alkyl having 1 to 4 carbon atoms, alkoxy having 1 to 4 carbon atoms, halogenoalkyl having 1 to 4 carbon atoms and 1 to 5 halogen atoms, halogenoalkoxy having 1 to 4 carbon atoms and 1 to 5 halogen atoms and halogenoalkylthio having 1 to 4 carbon atoms and 1 to 5 halogen atoms, ##STR4## R.sup.6 and R.sup.7 independently of one another each represent hydrogen or alkyl having 1 to 6 carbon atoms, 1 to 4 carbon atoms, phenyl, phenoxy, halogenoalkyl having 1 to 4 carbon atoms and 1 to 5 halogen atoms, halogenoalkoxy having 1 to 4 carbon atoms and 1 to 5 halogen atoms or represents halogenoalkylthio having 1 to 4 carbon atoms and 1 to 5 halogen atoms, and ##STR5## R.sup.8 and R.sup.9 independently of one another each represent hydrogen or alkyl having 1 to 6 carbon atoms, alkoxy having 1 to 4 carbon atoms, halogenoalkyl having 1 to 4 carbon atoms and 1 to 5 halogen atoms, halogenoalkoxy having 1 to 4 carbon atoms and 1 to 5 halogen atoms or phenyl, ##STR6## R.sup.10 represents alkyl having 1 to 6 carbon atoms, halogenoalkyl having 1 to 6 carbon atoms and 1 to 5 halogen atoms, cycloalkyl having 3 to 6 carbon atoms which is optionally substituted by halogen and/or alkyl having 1 to 4 carbon atoms, optionally substituted aryl or represents optionally substituted aralkyl, ##STR7## R.sup.11 represents hydrogen, alkyl or optionally substituted cycloalkyl, X.sup.3 represents halogen, alkyl having 1 to 4 carbon atoms, alkoxy having 1 to 4 carbon atoms, alkylthio having 1 to 4 carbon atoms, halogenoalkyl having 1 to 4 carbon atoms and 1 to 5 halogen atoms, halogenoalkoxy having 1 to 4 carbon atoms and 1 to 5 halogen atoms, halogenoalkylthio having 1 to 4 carbon atoms and 1 to 5 halogen atoms, phenyl which is optionally substituted by halogen and/or alkyl having 1 to 4 carbon atoms or represents phenoxy which is optionally substituted by halo-en and/or alkyl having 1 to 4 carbon atoms, ##STR8## R.sup.12 represents alkyl having 1 to 6 carbon atoms, halogenoalkyl having 1 to 4 carbon atoms and 1 to 5 halogen a
REFERENCES:
patent: 3912752 (1975-10-01), Meiser et al.
patent: 3952002 (1976-04-01), Kramer et al.
patent: 4048318 (1977-09-01), Meiser et al.
patent: 4079062 (1978-03-01), Van Reet et al.
patent: 4147791 (1979-04-01), Meiser et al.
patent: 4205075 (1980-05-01), Baldwin et al.
patent: 4243405 (1981-01-01), Balasubramanyan et al.
patent: 4464381 (1984-08-01), Janssen et al.
patent: 4532341 (1985-07-01), Holmwood et al.
patent: 4549900 (1985-10-01), Kramer et al.
patent: 4598085 (1986-07-01), Heeres et al.
patent: 4626595 (1986-12-01), Holmwood et al.
patent: 4652580 (1987-03-01), Janssen et al.
patent: 4723984 (1988-02-01), Holmwood et al.
patent: 4789672 (1988-12-01), Holmwood et al.
patent: 4871390 (1989-10-01), Holmwood et al.
patent: 4897107 (1990-01-01), Holmwood
patent: 4904297 (1990-02-01), Kramer et al.
patent: 4904298 (1990-02-01), Holmwood et al.
patent: 4906652 (1990-03-01), Karbach et al.
patent: 4911746 (1990-03-01), Holmwood et al.
patent: 4913727 (1990-04-01), Stroech et al.
patent: 4952232 (1990-08-01), Cuomo et al.
patent: 4965280 (1990-10-01), Cuomo et al.
patent: 4965281 (1990-10-01), Cuomo et al.
patent: 4968712 (1990-11-01), Elbe et al.
patent: 4980488 (1990-12-01), Stroech et al.
patent: 4988819 (1991-01-01), Stroech et al.
patent: 4990677 (1991-02-01), Stroech et al.
patent: 5034052 (1991-07-01), Stroech et al.
patent: 5081141 (1992-01-01), Colle et al.
patent: 5084465 (1992-01-01), Cuomo et al.
patent: 5087635 (1992-02-01), Shaber
patent: 5097047 (1992-03-01), Stroech et al.
patent: 5256683 (1993-10-01), Hutt et al.
patent: 5266585 (1993-11-01), Hubele et al.
patent: 5308743 (1994-05-01), Hutt et al.
patent: 5639918 (1997-06-01), Hutt et al.
patent: 5789430 (1998-08-01), Jautelat et al.
Piscopo et al, "Studies on heterocyclic compounds. etc" CA 99:194886 (1983).
Crom and Hammond, "Organic Chemistry", McGraw-Hill Book Co., NY (1964) 2nd ed., pp 565-567.
Dutzmann Stefan
Jautelat Manfred
Stenzel Klaus
Bayer Aktiengesellschaft
Gil Joseph C.
Marmo Carol
Morris Patricia L.
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