Acyl derivatives of 5-(2-(4-(1,2...

Details Acyl derivatives of 5-(2-(4-(1,2... Acyl derivatives of 5-(2-(4-(1,2...

2006-03-28

2006-03-28

Bernhardt, Emily (Department: 1624)

Drug, bio-affecting and body treating compositions

Designated organic active ingredient containing

Having -c-, wherein x is chalcogen, bonded directly to...

C544S368000

Reexamination Certificate

active

07019009

ABSTRACT:
A process for preparing acyl derivatives as prodrugs of 5-(2-(4-(1,2 benzisothiazole-3-yl)-1-piperazinyl)ethyl-6-chloro-1,3-dihydro-2H-indol-2-one and pharmaceutically acceptable acid addition salts and methods of use as an antipsychotic.

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patent: 0790236 (1997-08-01), None
patent: 0010975 (2000-03-01), None
Hans Bundgaard; Elsevier Science Publishers B.V.; Design of prodrugs: Bioreversible derivatives for various functional groups and chemical entities; (1985); p. 1-10.
Davis, et al.; CNS Drugs; Ziprazidone; (1997) vol. 8. No. 2; p. 153-159.
Caley, et al.; The Annals of Pharmacotherapy; Ziprasidone: The Atypical Antipsychotic; (2002) vol. 36, No. 5; p. 839-851.

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