Acid cleavable compounds, their preparation and use as bifunctio

Details Acid cleavable compounds, their preparation and use as bifunctio Acid cleavable compounds, their preparation and use as bifunctio

1993-03-04

1996-04-09

Tucker, Philip

Drug, bio-affecting and body treating compositions

Radionuclide or intended radionuclide containing; adjuvant...

549233, 549237, 549247, A61K 4300, C07D30760, C07D30794, C07D30789

Patent

active

055059317

ABSTRACT:
Novel compounds, their preparation and their use as bifunctional acid-labile crosslinking agents which are cleavable in an acid environment at a pH of below about 5.0 allowing for the controlled release of nucleophilic groups attached thereto are disclosed.

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