Acetamide derivatives

Drug – bio-affecting and body treating compositions – Designated organic active ingredient containing – Nitrogen containing other than solely as a nitrogen in an...

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514456, 514520, 514619, 514622, 514866, 549398, 549404, 549407, 558404, 558413, 564166, 564167, 564172, 564174, 564175, 564180, 564181, 564183, A61K 31165, C07C23357

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active

054300606

ABSTRACT:
The invention concerns novel N-phenylacetyl and related acyl derivatives of (4-amino-2,6-dimethylphenylsulphonyl)nitromethane and pharmaceutically acceptable salts thereof which are inhibitors of the enzyme aldose reductase and are of value, for example, in the treatment of certain peripheral effects of diabetes and galactosemia. Also disclosed are pharmaceutical compositions containing one of the derivatives and processes for the manufacture and use of the derivatives.

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