8a-AZA-8a-homoerythromycin cyclic iminoethers

Organic compounds -- part of the class 532-570 series – Organic compounds – Unsubstituted hydrocarbyl chain between the ring and the -c-...

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514183, 514450, A61K 3195, C07D52100

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active

051891590

ABSTRACT:
Cyclic iminoethers of the general structural formula wherein one of the R groups is hydrogen and the other R group represents a bond between the oxygen atom at C-6 or C-12 and the imino carbon at C-9; ##STR1## These compounds are macrolides useful as antibiotics and as intermediates for the synthesis of other macrolide antibiotics.

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