8-(5-Pyrimidinecarboxamide)nor-tropane derivatives

Details 8-(5-Pyrimidinecarboxamide)nor-tropane derivatives 8-(5-Pyrimidinecarboxamide)nor-tropane derivatives

1981-04-16

1982-03-23

Daus, Donald G.

Organic compounds -- part of the class 532-570 series

Organic compounds

Nitrogen attached directly or indirectly to the purine ring...

424251, 424265, 546124, 546125, C07D40114, A61K 31505

Patent

active

043213782

ABSTRACT:
There are disclosed nor-tropane derivatives substituted at the 3 position with aroylamino or heteroaroylamino and substituted at the 8 position with benzyl, substituted benzyl, 2-methyl thiophene, 3-methyl thiophene, 2-methyl furan or cyclohexylmethyl. The compounds are prepared by condensing the carboxylic acids corresponding to said aroyl or heteroaroyl group with the corresponding .beta.-3-amino-8-substituted nor-tropanes. The compounds possess neuroleptic properties.

REFERENCES:
patent: 3134782 (1964-05-01), Archer et al.
patent: 4179567 (1979-12-01), Clarke et al.
Ancher et al., "Chemical Abstracts", vol. 92, 1980, col. 58805g.

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