7-(substituted)cycloalkylamino-1 -(substituted)-6-fluoro-1,4-dih

Details 7-(substituted)cycloalkylamino-1 -(substituted)-6-fluoro-1,4-dih 7-(substituted)cycloalkylamino-1 -(substituted)-6-fluoro-1,4-dih

1990-02-01

1991-02-12

Shah, Mukund J.

Drug, bio-affecting and body treating compositions

Designated organic active ingredient containing

Having -c-, wherein x is chalcogen, bonded directly to...

546156, A61K 3147, C07D215333

Patent

active

049924494

ABSTRACT:
Novel antibacterial compounds of the formula: ##STR1## in which R.sub.1 is alkyl (C.sub.1 -C.sub.4), cycloalkyl (C.sub.3 -C.sub.6), alkoxy (C.sub.1 -C.sub.4), alkylamino (C.sub.1 -C.sub.3), vinyl, phenyl, benzyl, --CH.sub.2 CH.sub.2 F or mono or polysubstituted phenyl (wherein the substituent is halogen, CF.sub.3 or OCH.sub.2 F); n is an integer of from 1 to 4; and R.sub.2 is cis or trans hydroxy, amino, mono or disubstituted alkyl (C.sub.1 -C.sub.3) amino and the pharmacologically accepted salts thereof are described.

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