7-pyrrolyl tetracycline compounds and methods of use thereof

Details 7-pyrrolyl tetracycline compounds and methods of use thereof 7-pyrrolyl tetracycline compounds and methods of use thereof

2006-02-21

2006-02-21

Shameem, Golam M. M. (Department: 1626)

Drug, bio-affecting and body treating compositions

Designated organic active ingredient containing

Having -c-, wherein x is chalcogen, bonded directly to...

C514S381000, C514S399000, C514S406000, C548S255000, C548S529000, C552S203000, C552S204000, C552S205000

Reexamination Certificate

active

07001918

ABSTRACT:
A compound of Formula (I): wherein variables R, R1, R2, R3and A are as defined in the

REFERENCES:
patent: 2980584 (1961-04-01), Hammer
patent: 2990331 (1961-06-01), Neumann et al.
patent: 3062717 (1962-11-01), Hammer
patent: 3148212 (1964-09-01), Boothe et al.
patent: 3165531 (1965-01-01), Blackwood et al.
patent: 3226436 (1965-12-01), Petisi et al.
patent: RE26253 (1967-08-01), Petisi et al.
patent: 3338963 (1967-08-01), Petisi et al.
patent: 3341585 (1967-09-01), Bitha et al.
patent: 3345379 (1967-10-01), Martell
patent: 3345410 (1967-10-01), Winterbottom
patent: 3403179 (1968-09-01), Zambrano
patent: 3454697 (1969-07-01), Joyner et al.
patent: 3518306 (1970-06-01), Martell
patent: 3557260 (1971-01-01), Weber et al.
patent: 3579579 (1971-05-01), Hvalka et al.
patent: 3862225 (1975-01-01), Lloyd et al.
patent: 3901942 (1975-08-01), Bernardi et al.
patent: 3957980 (1976-05-01), Noseworthy
patent: 4018889 (1977-04-01), Armstrong
patent: 4024272 (1977-05-01), Rogalski et al.
patent: 4126680 (1978-11-01), Armstrong
patent: 5021407 (1991-06-01), Levy
patent: 5281628 (1994-01-01), Hlavka et al.
patent: 5284963 (1994-02-01), Sum et al.
patent: 5328902 (1994-07-01), Sum et al.
patent: 5380888 (1995-01-01), Sum et al.
patent: 5386041 (1995-01-01), Sum et al.
patent: 5401729 (1995-03-01), Sum et al.
patent: 5401863 (1995-03-01), Hlavka et al.
patent: 5420272 (1995-05-01), Sum et al.
patent: 5430162 (1995-07-01), Sum et al.
patent: 5457096 (1995-10-01), Sum et al.
patent: 5466684 (1995-11-01), Sum et al.
patent: 5494903 (1996-02-01), Hlavka et al.
patent: 5495018 (1996-02-01), Sum et al.
patent: 5495031 (1996-02-01), Sum et al.
patent: 5512553 (1996-04-01), Sum et al.
patent: 5530117 (1996-06-01), Hlavka et al.
patent: 5532227 (1996-07-01), Golub et al.
patent: 5789395 (1998-08-01), Amin et al.
patent: 5834450 (1998-11-01), Su
patent: 5886175 (1999-03-01), Sum et al.
patent: 6500812 (2002-12-01), Nelson et al.
patent: 6642270 (2003-11-01), Nelson et al.
patent: 6683068 (2004-01-01), Nelson et al.
patent: 6818634 (2004-11-01), Nelson et al.
patent: 6818635 (2004-11-01), Nelson et al.
patent: 2002/0128237 (2002-09-01), Nelson et al.
patent: 2004/0214800 (2004-10-01), Levy et al.
patent: 2004/0242548 (2004-12-01), Draper et al.
patent: 2005/0038002 (2005-02-01), Nelson et al.
patent: 0 536 346 (1993-04-01), None
patent: 0 536 515 (1993-04-01), None
patent: 0 582 788 (1994-02-01), None
patent: 0 582 789 (1994-02-01), None
patent: 0 582 790 (1994-02-01), None
patent: 0 582 810 (1994-02-01), None
patent: 1469384 (1977-04-01), None
patent: WO 00/28983 (2000-05-01), None
patent: WO 200204404 (2002-01-01), None
patent: WO 200204407 (2002-01-01), None
patent: WO 2004038000 (2004-05-01), None
patent: WO 2004038001 (2004-05-01), None
patent: WO 2004064728 (2004-08-01), None
patent: WO 2004091513 (2004-10-01), None
Koza, D. and Nsiah, Y., “Palladium catalyzed C-N Bond Formation in the Synthesis of 7-Amino-Substituted Tetracyclines,” J. Org. Chem., vol. 67, pp. 5025-5027 (2002), at p. 5026, 2nd col., compound 2f.
Koza, D. and Nsiah, Y., “Palladium Catalyzed C-N Bond Formation in the Synthesis of 7-Amino-Substituted Tetracyclines,” J. Org. Chem., vol. 67(14), pp. 5025-5027 (Jul. 2002), at p. 5026, Figure 1, compounds 2f, 2g, 2h, 2i.
Koza, D.J. “Synthesis of 7-substituted tetracycline derivatives,”Org. Lett.2(6):815-17 (2000).

Affiliated with

Also associated with

Rating

7-pyrrolyl tetracycline compounds and methods of use thereof does not yet have a rating. At this time, there are no reviews or comments for this patent.

If you have personal experience with 7-pyrrolyl tetracycline compounds and methods of use thereof, we encourage you to share that experience with our LandOfFree.com community. Your opinion is very important and 7-pyrrolyl tetracycline compounds and methods of use thereof will most certainly appreciate the feedback.

Rate now

Comments { 0 }

Profile ID: LFUS-PAI-O-3677817