7-azaindoles and the use thereof as therapeutic agents

Details 7-azaindoles and the use thereof as therapeutic agents 7-azaindoles and the use thereof as therapeutic agents

2011-05-24

2011-05-24

Davis, Zinna N (Department: 1625)

Drug, bio-affecting and body treating compositions

Designated organic active ingredient containing

Having -c-, wherein x is chalcogen, bonded directly to...

C514S337000, C546S113000, C546S278100

Reexamination Certificate

active

07947705

ABSTRACT:
The invention relates to substituted 7-azaindoles, process for their preparation, pharmaceutical preparations which comprise these compounds, and the pharmaceutical use of these compounds, which are inhibitors of phosphodiesterase 4, as active ingredients for the treatment of disorders which can be influenced by inhibition of phosphodiesterase 4 activity in particular in immunocompetent cells (e.g. macrophages and lymphocytes) by the compounds of the invention.

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