6-O-substituted macrolides having antibacterial activity

Details 6-O-substituted macrolides having antibacterial activity 6-O-substituted macrolides having antibacterial activity

1999-03-19

2000-04-25

Peselev, Elli

Drug, bio-affecting and body treating compositions

Designated organic active ingredient containing

Carbohydrate doai

536 72, 536 75, 536 185, A61K 3170, C07H 100, C07H 1708

Patent

active

06054435&

ABSTRACT:
The instant invention provides novel macrolide compounds and compositions useful in treating bacterial infections. Also provided are processes for preparing same.

REFERENCES:
patent: 5350839 (1994-09-01), Asaka et al.
patent: 5444051 (1995-08-01), Agouridas et al.
patent: 5527780 (1996-06-01), Agouridas et al.
patent: 5561118 (1996-10-01), Agouridas et al.
Pestka, et al. (I), "Effect of Erythromycin Analogues on Binding of [.sup.14 C] Erythromycin to Escherichia coli Ribosomes," Antimicrobial Agents and Chemotherapy, 6(4), 479-488 (Oct. 1974).
Pestka et al. (II), "Correlation of Effects of Erythromycin Analogues on Intact Bacteria and on [.sup.14 C] Erythromycin to Escherichia coli Ribosomes," Antimicrobial Agents and Chemotherapy, 6(4), 488-491 (Oct. 1974).
Pestka, et al. (III), "Inhibition of [.sup.14 C] Chloramphenicol Binding to Escherichia coli Ribosomes by Erythromycin Derivatives," Antimicrobial Agents and Chemotherapy, 6(1), 39-45 (Jul. 1974).
Pestka, et al. (IV), "Induction of Erythromycin Resistance in Staphylococcus aureus by Erythromycin Derivatives," Antimicrobial Agents and Chemotherapy, 9(1), 128-130 (Jan. 1976).
LeMahieu et al., "Glycoside Cleavage Reactions to Erythromycin A. Preparation of Erythromycin A." J. Medicinal Chem. 17 (9), 953-956 (Sep. 1974).

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