5-Substituted-2-phenylbenzo[b]thiophene-3-alkylamines and relate

Details 5-Substituted-2-phenylbenzo[b]thiophene-3-alkylamines and relate 5-Substituted-2-phenylbenzo[b]thiophene-3-alkylamines and relate

1977-09-26

1979-01-30

Coughlan, Jr., Paul M.

Organic compounds -- part of the class 532-570 series

Organic compounds

Nitrogen attached directly or indirectly to the purine ring...

2603265SA, 26032684, 2603305, C07D33358, C07D40906

Patent

active

041374142

ABSTRACT:
The invention encompasses novel 5-substituted-2-phenylbenzo[b]thiophene-3-alkylamines and related compounds of the general formula ##STR1## and the pharmaceutically acceptable acid addition salts thereof wherein R.sub.1 and R.sub.2 each independently represents H or an alkyl having from 1 to 8 carbon atoms or R.sub.1 and R.sub.2 together with N represents an azamonocyclic ring selected from the group comprising pyrrolidinyl, piperazinyl, substituted pyrrolidinyl wherein the substituent is an alkyl containing from 1 to 4 carbon atoms and substituted piperazinyl wherein the substituent is an alkyl containing from 1 to 4 carbon atoms or an alkanol wherein the alkyl moiety contains 1 to 4 carbon atoms; Y represents H, halogen or alkyl having 1 to 4 carbon atoms; X represents H, halogen, alkyl having 1 to 4 carbon atoms and alkoxy wherein the alkyl moiety contains 1 to 4 carbon atoms; and n is a positive integer from 1 to 4. These compounds possess utility as neuroleptics or anti-bacterial agents.

REFERENCES:
patent: 3070606 (1962-12-01), Anderson
patent: 3594478 (1971-07-01), Brandstrom et al.
patent: 3910955 (1975-10-01), Chapman et al.
patent: 3947470 (1976-03-01), Brenner et al.
Descamps et al, Chim. Ther., vol. 8 (1973), pp. 536-544.

Affiliated with

Also associated with

Rating

5-Substituted-2-phenylbenzo[b]thiophene-3-alkylamines and relate does not yet have a rating. At this time, there are no reviews or comments for this patent.

If you have personal experience with 5-Substituted-2-phenylbenzo[b]thiophene-3-alkylamines and relate, we encourage you to share that experience with our LandOfFree.com community. Your opinion is very important and 5-Substituted-2-phenylbenzo[b]thiophene-3-alkylamines and relate will most certainly appreciate the feedback.

Rate now

Comments { 0 }

Profile ID: LFUS-PAI-O-1151485