5-phenylpyrimidines, their preparation, compositions...

Drug – bio-affecting and body treating compositions – Designated organic active ingredient containing – Having -c- – wherein x is chalcogen – bonded directly to...

Reexamination Certificate

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C514S269000, C514S272000, C514S275000, C544S326000, C544S334000, C544S317000, C544S320000, C544S325000

Reexamination Certificate

active

07449471

ABSTRACT:
5-Phenylpyrimidines of the formula Iin which the substituents and the index are as defined below:R1,R2are hydrogen, alkyl, haloalkyl, cycloalkyl, halocycloalkyl, alkenyl, haloalkenyl, alkynyl or haloalkynyl, and R1and R2together with the nitrogen atom to which they are attached may also form a saturated or unsaturated ring which may be interrupted by an ether, thio, sulfoxyl or sulfonyl group and may be substituted by one to four groups Raand/or Rb;R3is hydrogen, halogen, cyano, alkyl, haloalkyl, alkoxy, haloalkoxy or alkenyloxy;R4is hydrogen, halogen, cyano, hydroxyl, mercapto, azido, alkyl, alkenyl, alkynyl, haloalkyl, alkoxy, alkenyloxy, alkynyloxy, haloalkoxy, alkylthio, alkenylthio, alkynylthio, haloalkylthio, —ON═CRaRb, —CRc═NORa, —NRcN═CRaRb, —NRaRb, —NRcNRaRb, —NORa, —NRcC(═NRc′)NRaRb, —NRcC(═O)NRaRb, —NRaC(═O)Rc, —NRaC(═NORc)Rc′, —OC(═O)Rc, —C(═NORc)NRaRb, —CRc(═NNRaRb), —C (═O)NRaRbor —C(═O)Rc;in which Ra, Rband Rcare as defined in the description;X is halogen, alkyl, alkoxy or haloalkyl; andm is an integer from 1 to 5 ;processes for preparing these compounds, compositions comprising them and their use for controlling harmful fungi are described.

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