5-modified pyrimidines from palladium catalyzed carbon-carbon co

Details 5-modified pyrimidines from palladium catalyzed carbon-carbon co 5-modified pyrimidines from palladium catalyzed carbon-carbon co

1995-04-19

1997-01-07

Wilson, James O.

Organic compounds -- part of the class 532-570 series

Organic compounds

Carbohydrates or derivatives

536 281, 536 284, 536 285, 536 2851, 536 2853, 536 2854, C07H 100, C07H 1900

Patent

active

055918433

ABSTRACT:
This invention discloses a method for the preparation of pyrimidine nucleosides modified at the 5-position of the pyrimidine ring using a palladium catalyst of the formula PdL.sub.3, wherein L is a ligand of palladium. Included in the invention are pyrimidine nucleosides modified at the 5-position prepared according to the method of the invention.

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