5-lipoxygenase-activating protein (FLAP) inhibitors

Drug – bio-affecting and body treating compositions – Designated organic active ingredient containing – Having -c- – wherein x is chalcogen – bonded directly to...

Reexamination Certificate

Rate now

  [ 0.00 ] – not rated yet Voters 0   Comments 0

Details

C546S277400, C546S277700, C548S484000, C548S490000, C514S418000

Reexamination Certificate

active

07834037

ABSTRACT:
Described herein are compounds and pharmaceutical compositions containing such compounds, which modulate the activity of 5-lipoxygenase-activating protein (FLAP). Also described herein are methods of using such FLAP modulators, alone and in combination with other compounds, for treating respiratory, cardiovascular, and other leukotriene-dependent or leukotriene mediated conditions or diseases.

REFERENCES:
patent: 4273782 (1981-06-01), Cross et al.
patent: 4616009 (1986-10-01), Tahara et al.
patent: 4826987 (1989-05-01), Nielsen et al.
patent: 5081138 (1992-01-01), Gillard et al.
patent: 5081145 (1992-01-01), Guindon et al.
patent: 5093356 (1992-03-01), Girard et al.
patent: 5095031 (1992-03-01), Brooks et al.
patent: 5109009 (1992-04-01), Nielsen et al.
patent: 5157039 (1992-10-01), Nielsen et al.
patent: 5182367 (1993-01-01), Gillard et al.
patent: 5190968 (1993-03-01), Gillard et al.
patent: 5202321 (1993-04-01), Hutchinson et al.
patent: 5204344 (1993-04-01), Prasit et al.
patent: 5225421 (1993-07-01), Gillard et al.
patent: 5229516 (1993-07-01), Musser et al.
patent: 5232916 (1993-08-01), Zamboni et al.
patent: 5252585 (1993-10-01), Frenette et al.
patent: 5254567 (1993-10-01), Down et al.
patent: 5272145 (1993-12-01), Prasit et al.
patent: 5273980 (1993-12-01), Frenette et al.
patent: 5288743 (1994-02-01), Brooks et al.
patent: 5290788 (1994-03-01), Stevens et al.
patent: 5290798 (1994-03-01), Gillard et al.
patent: 5308850 (1994-05-01), Gillard et al.
patent: 5314898 (1994-05-01), Chung et al.
patent: 5334719 (1994-08-01), Frenette
patent: 5374635 (1994-12-01), Leger et al.
patent: 5380850 (1995-01-01), Prasit et al.
patent: 5389650 (1995-02-01), Frenette et al.
patent: 5399699 (1995-03-01), Kolasa et al.
patent: 5420282 (1995-05-01), Brooks et al.
patent: 5420289 (1995-05-01), Musser et al.
patent: 5459150 (1995-10-01), Brooks et al.
patent: 5635516 (1997-06-01), Caubere et al.
patent: 5750558 (1998-05-01), Brooks et al.
patent: 5877329 (1999-03-01), Chen et al.
patent: 5972241 (1999-10-01), Johnson et al.
patent: 6246452 (2001-06-01), Sekine et al.
patent: 6500853 (2002-12-01), Seehra et al.
patent: 6855722 (2005-02-01), Lu et al.
patent: 7118869 (2006-10-01), Blumenfeld et al.
patent: 7405302 (2008-07-01), Hutchinson et al.
patent: 2001/0039037 (2001-11-01), Harland
patent: 2003/0203833 (2003-10-01), Ignar et al.
patent: 2004/0014759 (2004-01-01), Picard et al.
patent: 2004/0086952 (2004-05-01), Gentz et al.
patent: 2004/0198800 (2004-10-01), Allan et al.
patent: 2005/0245515 (2005-11-01), Dehmlow et al.
patent: 2006/0211677 (2006-09-01), Chu et al.
patent: 2007/0003971 (2007-01-01), Blumenfeld et al.
patent: 2007/0105866 (2007-05-01), Hutchinson et al.
patent: 2007/0123522 (2007-05-01), Hutchinson et al.
patent: 2007/0219206 (2007-09-01), Hutchinson et al.
patent: 2007/0225285 (2007-09-01), Hutchinson et al.
patent: 2007/0244128 (2007-10-01), Hutchinson et al.
patent: 2008/0227807 (2008-09-01), Hutchinson et al.
patent: 2008/0293739 (2008-11-01), Trede
patent: 2009/0018170 (2009-01-01), Hutchinson et al.
patent: 2032253 (1991-06-01), None
patent: 1337427 (1995-10-01), None
patent: 4338770 (1995-05-01), None
patent: 0510398 (1992-10-01), None
patent: 0535924 (1993-04-01), None
patent: 0540051 (1993-05-01), None
patent: 0597112 (1994-05-01), None
patent: 0419049 (1995-04-01), None
patent: 2280181 (1995-01-01), None
patent: 6058881 (1994-03-01), None
patent: 6100551 (1994-04-01), None
patent: 7005651 (1995-01-01), None
patent: 08020532 (1996-01-01), None
patent: 09002977 (1997-01-01), None
patent: 11080032 (1999-03-01), None
patent: 11189531 (1999-07-01), None
patent: 11193265 (1999-07-01), None
patent: 2000007590 (2000-01-01), None
patent: 2000302671 (2000-10-01), None
patent: 2001139462 (2001-05-01), None
patent: 2002226429 (2002-08-01), None
patent: 3457694 (2003-08-01), None
patent: 2005082701 (2005-03-01), None
patent: 2005170939 (2005-06-01), None
patent: 2005194250 (2005-07-01), None
patent: 8802364 (1988-04-01), None
patent: WO-91-06537 (1991-05-01), None
patent: 9203132 (1992-03-01), None
patent: WO-93-16069 (1993-08-01), None
patent: WO-93-20065 (1993-10-01), None
patent: 9323391 (1993-11-01), None
patent: WO-93-25546 (1993-12-01), None
patent: 9400446 (1994-01-01), None
patent: 9411378 (1994-05-01), None
patent: 9412179 (1994-06-01), None
patent: 9413293 (1994-06-01), None
patent: 9413662 (1994-06-01), None
patent: 9429290 (1994-12-01), None
patent: 9506637 (1995-03-01), None
patent: 9535372 (1995-12-01), None
patent: 9603377 (1996-02-01), None
patent: 9615118 (1996-05-01), None
patent: WO-96-18393 (1996-06-01), None
patent: WO-96-32379 (1996-10-01), None
patent: 9635670 (1996-11-01), None
patent: 9728105 (1997-08-01), None
patent: WO-97-41100 (1997-11-01), None
patent: 9749703 (1997-12-01), None
patent: 9803202 (1998-01-01), None
patent: 9821184 (1998-05-01), None
patent: 9852943 (1998-11-01), None
patent: 9856757 (1998-12-01), None
patent: 9933458 (1999-07-01), None
patent: WO-99-33800 (1999-07-01), None
patent: 9943651 (1999-09-01), None
patent: 9943672 (1999-09-01), None
patent: 9952942 (1999-10-01), None
patent: 0029574 (2000-05-01), None
patent: 0043384 (2000-07-01), None
patent: 0144184 (2000-12-01), None
patent: 0121594 (2001-03-01), None
patent: 0132621 (2001-05-01), None
patent: 0136403 (2001-05-01), None
patent: 0141807 (2001-06-01), None
patent: 0159105 (2001-08-01), None
patent: WO-01-58869 (2001-08-01), None
patent: 0164639 (2001-09-01), None
patent: 0166520 (2001-09-01), None
patent: 0170211 (2001-09-01), None
patent: 0177149 (2001-10-01), None
patent: 0200621 (2002-01-01), None
patent: 0210152 (2002-02-01), None
patent: 0228835 (2002-04-01), None
patent: 02051397 (2002-07-01), None
patent: 02051837 (2002-07-01), None
patent: 03022813 (2003-03-01), None
patent: 03022814 (2003-03-01), None
patent: 03028719 (2003-04-01), None
patent: 03035625 (2003-05-01), None
patent: WO 03-044014 (2003-05-01), None
patent: 03050174 (2003-06-01), None
patent: 03094889 (2003-11-01), None
patent: 03099771 (2003-12-01), None
patent: 2004000795 (2003-12-01), None
patent: WO-2004-000831 (2003-12-01), None
patent: 2004017917 (2004-03-01), None
patent: 2004017920 (2004-03-01), None
patent: 2004043392 (2004-05-01), None
patent: 2004048331 (2004-06-01), None
patent: 2004050643 (2004-06-01), None
patent: 2004065388 (2004-08-01), None
patent: 2004078719 (2004-09-01), None
patent: 2004101554 (2004-11-01), None
patent: 2004108671 (2004-12-01), None
patent: 2005009951 (2005-02-01), None
patent: 2005019381 (2005-03-01), None
patent: 2005023246 (2005-03-01), None
patent: 2005023806 (2005-03-01), None
patent: WO-2005-030717 (2005-04-01), None
patent: 2005054193 (2005-06-01), None
patent: 2005065266 (2005-07-01), None
patent: 2005066151 (2005-07-01), None
patent: 2005066157 (2005-07-01), None
patent: 2005082346 (2005-09-01), None
patent: 2005097203 (2005-10-01), None
patent: 2005112921 (2005-12-01), None
patent: 2005123674 (2005-12-01), None
patent: WO-2006-014262 (2006-02-01), None
patent: 2006023843 (2006-03-01), None
patent: 2006030031 (2006-03-01), None
patent: 2006044602 (2006-04-01), None
patent: 2006074984 (2006-07-01), None
patent: 2006077364 (2006-07-01), None
patent: 2006077365 (2006-07-01), None
patent: 2006077366 (2006-07-01), None
patent: 2006077367 (2006-07-01), None
patent: 2006098912 (2006-09-01), None
patent: 2006105439 (2006-10-01), None
patent: WO-2006-111560 (2006-10-01), None
patent: 2006131737 (2006-12-01), None
patent: 2007022427 (2007-02-01), None
patent: 2007048042 (2007-04-01), None
patent: WO-2007-047204 (2007-04-01), None
patent: WO-2007-047207 (2007-04-01), None
patent: WO-2007-056021 (2007-05-01), None
patent: WO-2007-056220 (2007-05-01), None
patent: WO-2007-056228 (2007-05-01), None
patent: 2007109279 (2007-09-01), None
patent: 2007123225 (2007-11-01), None
patent: 2008058341 (2008-05-01), None
patent: 2008067566 (2008-06-01), None
patent: 2008097930 (2008-08-01), None
patent: 2008127728 (2008-10-01), None
patent: WO-2008-137609 (2008-11-01), None
patent: WO-2008-137805 (2008-11-01), None
patent: WO-2008-141011 (2008-11-01), None
patent: 200900274

LandOfFree

Say what you really think

Search LandOfFree.com for the USA inventors and patents. Rate them and share your experience with other people.

Rating

5-lipoxygenase-activating protein (FLAP) inhibitors does not yet have a rating. At this time, there are no reviews or comments for this patent.

If you have personal experience with 5-lipoxygenase-activating protein (FLAP) inhibitors, we encourage you to share that experience with our LandOfFree.com community. Your opinion is very important and 5-lipoxygenase-activating protein (FLAP) inhibitors will most certainly appreciate the feedback.

Rate now

     

Profile ID: LFUS-PAI-O-4211541

  Search
All data on this website is collected from public sources. Our data reflects the most accurate information available at the time of publication.