5-HT 7 receptor antagonists

Drug – bio-affecting and body treating compositions – Designated organic active ingredient containing – Having -c- – wherein x is chalcogen – bonded directly to...

Reexamination Certificate

Rate now

  [ 0.00 ] – not rated yet Voters 0   Comments 0

Details

C546S139000

Reexamination Certificate

active

10920738

ABSTRACT:
The invention relates to compounds having pharmacological activity towards the 5-HT7 receptor, and more particularly to some tetrahydroisoquinoline substituted sulfonamide compounds, to processes of preparation of such compounds, to pharmaceutical compositions comprising them, and to their use for the treatment and or prophylaxis of a disease in which 5-HT is involved, such as CNS disorders.

REFERENCES:
patent: 5294621 (1994-03-01), Russell
patent: 0 021 580 (1983-12-01), None
patent: 0 076 072 (1987-05-01), None
patent: WO 97/29097 (1997-08-01), None
patent: WO 97/48681 (1997-12-01), None
patent: WO 97/49695 (1997-12-01), None
patent: WO 99/24022 (1999-05-01), None
patent: WO 00/00472 (2000-01-01), None
patent: WO 03/037887 (2003-05-01), None
patent: WO 03/048118 (2003-06-01), None
Yamazaki et al, Chemical Abstracts, vol. 54, Abstracts 28777, 1960.
Vermeulen et al, J. Med. Chem, vol. 47, pp. 5451-5466, Sep. 2004.
Yamazaki et al, vol. 79, pp. 1014-1018, 1960, English Language Translation.
Terron, J. A., IDrugs, vol. 1(3), pp. 302-301, 1998.
Lovenberg et al., Neuron, vol. 11, pp. 449-458, 1993.
Terron, J. A., Br. J. Pharmacol., vol. 121, pp. 563-571, 1997.
Schoeffter et al., Br. J. Pharmacol., vol. 117, pp. 993-994, 1996.
Terron, J. A., Eur. J. Pharmacol., vol. 439, pp. 1-11, 2002.
De Ponti et al., Drugs, vol. 61, pp. 317-332, 2001.
Read et al., Br. J. Pharmacol., vol. 140, pp. 53-60, Jul. 29, 2003.
Wesolowska, A., Polish J. Pharmacol., vol. 54, pp. 327-341, 2002.
Mokrosz et al., J. Med. Chem., vol. 39, pp. 1125-1129, 1996.
Contreras et al., J. Med. Chem., vol. 42, pp. 730-741, 1999.
Alvarez et al., J. Med. Chem., vol. 30, pp. 1186-1193, 1987.
Alvarez et al., Anales Quimica, vol. 80, pp. 283-290, 1984.
Austin et al., Bioorg. Med. Chem. Lett., vol. 9, pp. 179-184, 1999.
Greene et al., Protective Groups in Organic Synthesis, 3rdEd., John Wiley & Sons, Inc., pp. v, xi, xii, 1999.
Mach et al., Bioorg. Med. Chem. Lett., vol. 14(1), pp. 195-202, Jan. 5, 2004.
Munson et al., Anal. Biochem., vol. 107, pp. 220-239, 1980.
Bon et al., J. Org. Chem., vol. 59, pp. 1904-1906, 1994.
European Patent Office, European Search Report for EP 04380171.1, issued Jan. 25, 2005.
Zhu et al., J. Med. Chem., vol. 46, pp. 831-837, Jan. 21, 2003.

LandOfFree

Say what you really think

Search LandOfFree.com for the USA inventors and patents. Rate them and share your experience with other people.

Rating

5-HT 7 receptor antagonists does not yet have a rating. At this time, there are no reviews or comments for this patent.

If you have personal experience with 5-HT 7 receptor antagonists, we encourage you to share that experience with our LandOfFree.com community. Your opinion is very important and 5-HT 7 receptor antagonists will most certainly appreciate the feedback.

Rate now

     

Profile ID: LFUS-PAI-O-3810126

  Search
All data on this website is collected from public sources. Our data reflects the most accurate information available at the time of publication.