5,11-dihyro-6H-dipyrido[3,2-B:2',3'-e][1,3]diazepines and their

Details 5,11-dihyro-6H-dipyrido[3,2-B:2',3'-e][1,3]diazepines and their 5,11-dihyro-6H-dipyrido[3,2-B:2',3'-e][1,3]diazepines and their

1994-07-22

1997-04-15

Bond, Robert T.

Drug, bio-affecting and body treating compositions

Designated organic active ingredient containing

Heterocyclic carbon compounds containing a hetero ring...

540495, 540557, A61K 3155, C07D47114

Patent

active

056209746

ABSTRACT:
Disclosed are novel 5,11-dihydro-6H-dipyrido[3,2-b; 2',3'-e][1,4]diazepines. These are useful in the prevention or treatment of HIV infection.

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Chemical Abstracts, vol. 90, No. 17 1979, abstracting Thoma-GmbH 11 Substituted 5,11-dihydro-6H-pyrido-[2,3-b][1,4]benzo-diazepine-6-ones, p. 522, col. 1, abstract No. 90:1378875s.
Chemical Abstracts vol. 90, No. 19 1979, p. 611, Col. 2, Abstract No. 90,152145x abstracting Brewster et al.
The Synthosis of some pyrido [1,4]benzoxazepines and dipyrido [1,4]oxzepines.
Chemical Abstracts, vol. 71, No. 23 (1964) p. 394, Col. 1 abstract No. 90:112,994, abstracting Schmidt et al. "Analgesic 5,11-dihydro-6-H-pyrido[2,3-b][1,4]benzo-diazepines-6-ones".
Hargrave et al., "Novel Non-Nucleoside Inhibitors of HIV-1 Reverse Transcriptase, Tricyclic Pyrido benzo-and Dipyridodiazepines" J. Med. Chem. (1991) vol. 34 pp. 2231-2241.
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Koup et al. "Inhibition of Human Immunodeficiency Virus Type 1 (HIV-1) Replication by the Dipyridodiazepinone BI-RG-587" The Journal of Infectious Diseases (191) vol. 163 pp. 466-470.
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