4-piperazinyl benzenesulfonyl indoles and uses thereof

Details 4-piperazinyl benzenesulfonyl indoles and uses thereof 4-piperazinyl benzenesulfonyl indoles and uses thereof

2006-04-04

2006-04-04

Bernhardt, Emily (Department: 1624)

Drug, bio-affecting and body treating compositions

Designated organic active ingredient containing

Having -c-, wherein x is chalcogen, bonded directly to...

C544S373000

Reexamination Certificate

active

07022708

ABSTRACT:
This invention relates to compounds which have generally 5-HT6 receptor affinity and which are represented by Formula I:wherein R1, R2, R3, R4, and R5are as defined herein; or individual isomers, racemic or non-racemic mixtures of isomers, or pharmaceutically acceptable salts or solvates thereof. The invention further relates to pharmaceutical compositions containing such compounds, methods for their use as therapeutic agents, and methods of preparation thereof.

REFERENCES:
patent: 2004/0024210 (2004-02-01), Johanssen et al.
patent: 2 729 144 (1996-07-01), None
patent: WO 93/03012 (1993-02-01), None
patent: WO 98/27081 (1998-06-01), None
patent: WO 99/02502 (1999-01-01), None
patent: WO 00/58304 (2000-10-01), None
patent: WO 01/64642 (2001-09-01), None
patent: WO 03/104193 (2003-12-01), None
Robichaud et al. in Annual Reports in Medicinal Chemistry, vol. 36, p. 11-20 (2000).
Rogers et al. Psychopharmacology, vol. 158, p. 114-119 (2001).
Bromidge et al. Bioorganic & Medicinal Chemistry Letters, vol. 11, p. 55-58 (2001).

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