Drug – bio-affecting and body treating compositions – Designated organic active ingredient containing – Heterocyclic carbon compounds containing a hetero ring...
Reexamination Certificate
2005-12-13
2005-12-13
Stockton, Laura L. (Department: 1626)
Drug, bio-affecting and body treating compositions
Designated organic active ingredient containing
Heterocyclic carbon compounds containing a hetero ring...
C514S326000, C514S403000, C544S140000, C546S211000, C548S379400
Reexamination Certificate
active
06974810
ABSTRACT:
The present invention relates to a group of novel 4,5-dihydro-1H-pyrazole derivatives which are potent cannabinoid (CB1) receptor antagonists with utility for the treatment of diseases connected with disorders of the cannabinoid system. The compounds have the general formula (Ia) or (Ib) wherein the symbols have the meanings given in the specification. The invention also relates to methods for the preparation of these compounds, and to pharmaceutical compositions containing one or more of these compounds as an active component
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Jochen Antel et al., “Novel Medical Uses of Compounds Showing CB1-Antagonistic Activity and Combination Treatment Involving Said Compounds,” US-10/969,840, filed on Oct. 22, 2004.
Jochen Antel et al., “Novel Medical Combination Treatment of Obesity Involving 4,5-Dihydro-1H-Pyrazole Derivatives Having CB1-Antagonistic Activity,” US-10/972,006, filed on Oct. 25, 2004.
Jochen Antel et al., “Novel Medical Combination Treatment of Obesity Involving 4,5-Dihydro-1H-Pyrazole Derivatives Having CB1-Antagonistic Activity,” US-11/005,486, filed on Dec. 7, 2004.
Herremans Arnoldus H. J.
Kruse Cornelis G.
Lange Josephus H. M.
Stuivenberg Herman H. van
Tipker Jacobus
Finnegan Henderson Farabow Garrett & Dunner L.L.P.
Solvay Pharmaceuticals B.V.
Stockton Laura L.
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