3-substituted-aminomethyl-3-subs tituted-oxy-17A-methyl-17A-lowe

Details 3-substituted-aminomethyl-3-subs tituted-oxy-17A-methyl-17A-lowe 3-substituted-aminomethyl-3-subs tituted-oxy-17A-methyl-17A-lowe

1992-06-08

1993-07-20

Daus, Donald G.

Organic compounds -- part of the class 532-570 series

Organic compounds

Unsubstituted hydrocarbyl chain between the ring and the -c-...

546 77, 544125, 544361, C07J 7300

Patent

active

052295117

ABSTRACT:
This invention pertains to novel 3-substituted-aminomethyl-3-substituted-oxy-17a-methyl-17a-lower-alkyl-17a -aza-D-homo-5-alpha-androstane compounds useful as muscle relaxants, methods for preparing such compounds, and method for administering muscle relaxation, wherein the novel compounds are represented the general formula: ##STR1## including optical active isomeric forms, and pharmaceutically acceptable acid addition salts thereof, wherein:

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