3-O-glycosyl 16-membered macrolide antibacterials and related de

Drug – bio-affecting and body treating compositions – Designated organic active ingredient containing – Carbohydrate doai

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536 71, A61K 3170, C07H 1708

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049621467

ABSTRACT:
3-O-Glycosyl derivatives of 16-membered macrolides such as O-.alpha.-L-cladinosyl-(1.fwdarw.3)-12,13-dehydro-12,13-deoxorosaramicin, 2", 4",4'"-tri-O-acetyl-O-(4'-O-phenoxyacetyl-.alpha.-L-cladinosyl)-(1.fwdarw. 3)-desmyconsin and pharmaceutically acceptable acid addition salts thereof useful as antibacterials are disclosed.

REFERENCES:
patent: 3178341 (1965-04-01), Hamill et al.
patent: 3326759 (1967-06-01), Hamill et al.
patent: 3769273 (1973-10-01), Massey
patent: 3975372 (1976-08-01), Ganguly et al.
patent: 4056616 (1977-11-01), Reimann et al.
patent: 4161523 (1979-07-01), Weinstein et al.
patent: 4234690 (1980-11-01), Weinstein et al.
patent: 4252898 (1981-02-01), Nash et al.
patent: 4321361 (1982-03-01), Baltz et al.
patent: 4345069 (1982-08-01), Sakakibara et al.
patent: 4357325 (1982-11-01), Ose et al.
patent: 4415730 (1983-11-01), Fujiwara et al.
patent: 4454314 (1984-06-01), Nagel
patent: 4477443 (1984-10-01), Umezawa et al.
patent: 4528369 (1985-07-01), Wild
Chemical Abstracts, vol. 102, (No. 15), Apr. 15, 1985, Abstract No. 132421x.
Chemical Abstracts, vol. 108, (No. 19), Sep. 9, 1987, Abstract No. 167885c.
Djerassi et al., J. Am. Chem. Soc., 1956, vol. 78, pp. 6390-6395.
Wiley et al., J. Am. Chem. Soc., 1957, vol. 79, pp. 6062-6072.
Djerassi et al., Tetrahedron, 1958, vol. 3, pp. 255-268.
Straustz et al., J. Am. Chem. Soc., 1960, vol. 82, pp. 3225-3227.
Egan et al., J. Am. Chem. Soc., 1970, vol. 92, pp. 4129-4130.
Pigman et al., The Carbohydrates, Academic Press., 2nd Ed., 1980, pp. 767-798.
Brimacombe et al., J. Chem. Soc., Perkin Trans. I, 1982, pp. 2583-2587.

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