Drug – bio-affecting and body treating compositions – Designated organic active ingredient containing – Having -c- – wherein x is chalcogen – bonded directly to...
Patent
1984-07-30
1986-06-10
Love, Ethel G.
Drug, bio-affecting and body treating compositions
Designated organic active ingredient containing
Having -c-, wherein x is chalcogen, bonded directly to...
544277, C07D47300, A61K 3152
Patent
active
045943508
ABSTRACT:
Antiviral (3-ethoxypropionate) esters of (+)-cyclaradine having the formula: ##STR1## In the monoester Ry and Rz are hydrogen. In the diester Ry is the 3-ethoxypropionyl group and Rz is hydrogen. In the triester, Ry and Rz are each 3-ethoxypropionyl groups.
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Shannon, W. et al., Antimicrob. Agents and Chemother., (1983), 24, pp. 538-543; Comparison of the Efficacy of Vidarabine, its carbocyclic Analog (Cyclaradine), and Cylaradine-5'-Methoxyacetate in the Treatment of Herpes.
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Hoffman Thomas
Love Ethel G.
Reagents of University of Minnesota
Rosen Gerald S.
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