3'-azido-2',3'-dideoxy-5-methylcytidine anti-viral composition

Details 3'-azido-2',3'-dideoxy-5-methylcytidine anti-viral composition 3'-azido-2',3'-dideoxy-5-methylcytidine anti-viral composition

1990-06-06

1991-12-31

Rollins, John W.

Drug, bio-affecting and body treating compositions

Designated organic active ingredient containing

Carbohydrate doai

514 51, A61K 3170

Patent

active

050772791

ABSTRACT:
A composition delivering an HIV-inhibitory amount of an active compound of the general formula: ##STR1## wherein R is OH, monophosphate, diphosphate, or triphosphate, or a pharmacologically acceptable salt thereof; and wherein the means is a pharmaceutically acceptable carrier. In the preferred embodiment, an effective dose of 3'-azido-2',3'-dideoxy-5-methylcytidine, or its derivatives, is administered in a pharmaceutically acceptable carrier to a patient for the treatment of AIDS.

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